γ-Carboline Synthesis by Heterocyclization of TosMIC Derivatives

The Journal of Organic Chemistry
Sara GutiérrezJuan J Vaquero

Abstract

A new method for the synthesis of γ-carbolines by a heterocyclization that involves α-indol-2-ylmethyl TosMIC derivatives and different electrophiles has been developed. This methodology has been successfully applied to the synthesis of several highly substituted γ-carbolines.

References

Jun 30, 2001·The Journal of Organic Chemistry·J D FreedN A Magomedov
Jun 4, 2005·The Journal of Organic Chemistry·Alejandro BaezaJuan J Vaquero
Jul 14, 2006·Chemical Reviews·Guy R Humphrey, Jeffrey T Kuethe
Feb 20, 2007·Current Medicinal Chemistry·Rihui CaoAnlong Xu
Nov 6, 2010·Angewandte Chemie·Alexander V Lygin, Armin de Meijere
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Mar 16, 2017·Angewandte Chemie·Sergiy V ChepyshevFraser F Fleming
Nov 29, 2017·The Journal of Organic Chemistry·Anthony Y ChenHaiming Zhang

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Citations

Jun 30, 2019·Organic & Biomolecular Chemistry·Arun Divakar Mathiyazhagan, Gopinathan Anilkumar
Jul 6, 2021·Beilstein Journal of Organic Chemistry·Premansh DudheVenkatesh Chelvam
Jun 15, 2019·Organic Letters·Shalini VermaAkhilesh K Verma
Dec 7, 2021·The Journal of Organic Chemistry·Masahiro AkitakeShinji Tanimori

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