N-Arylations of trifluoromethylated N-acylhydrazones with diaryliodonium salts as arylation reagents

Organic & Biomolecular Chemistry
Huaiyuan ZhangYulai Hu

Abstract

A novel and efficient N-arylation of trifluoromethylated N-acylhydrazones is described by using diaryliodonium salts as arylation reagents in the presence of copper salts. A wide variety of N-aryl acylhydrazones are obtained with good to excellent yields under mild reaction conditions.

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Citations

Oct 16, 2019·Mini Reviews in Medicinal Chemistry·Juliana de Oliveira Carneiro BrumJosé Daniel Figueroa Villar

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Methods Mentioned

BETA
silica

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