Reaction of arynes with amino acid esters

Chemical Communications : Chem Comm
Kentaro OkumaYoshinobu Yokomori

Abstract

An efficient route to a variety of 2-phenylindolin-3-ones from amino acid methyl esters has been developed. The reaction of amino acid methyl esters with benzyne prepared from 2-(trimethylsilyl)phenyl triflate and CsF gave 2-phenylindolin-3-ones in moderate to good yields.

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Citations

Feb 24, 2012·The Journal of Organic Chemistry·Donald C RognessRichard C Larock
Apr 9, 2016·The Journal of Organic Chemistry·Lanlan ZhangZhong Jin
Jun 16, 2016·Organic Letters·Dachuan QiuYang Li
Mar 14, 2018·Chemistry : a European Journal·Hortense LauwickMathieu Achard
Jul 6, 2012·Chemistry : a European Journal·Chepuri V Suneel KumarChepuri V Ramana
Aug 22, 2013·Organic & Biomolecular Chemistry·Jaya Kishore VandavasiJeh-Jeng Wang
Nov 8, 2012·Organic & Biomolecular Chemistry·Anton V DubrovskiyRichard C Larock
Apr 13, 2013·Chemical Communications : Chem Comm·Yogesh Goriya, Chepuri V Ramana
Feb 19, 2021·Chemical Reviews·Jiarong ShiYang Li
Mar 15, 2012·The Journal of Organic Chemistry·Pan LiFeng Shi
Dec 17, 2014·The Journal of Organic Chemistry·Charles E Hendrick, Qiu Wang
Apr 17, 2015·Journal of the American Chemical Society·Jiarong ShiYang Li
Jun 16, 2011·Organic Letters·Donald McAuslandMichael F Greaney
Aug 24, 2011·Organic Letters·Kallolmay Biswas, Michael F Greaney

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