Regioselective Ir(III)-catalyzed C-H alkynylation directed by 7-azaindoles

Organic & Biomolecular Chemistry
Bin LiuRuntao Li

Abstract

Herein we report a novel iridium(iii)-catalyzed ortho-mono-alkynylation of 7-azaindoles under mild conditions. This approach provides a general and straightforward access to form novel 7-azaindole derivatives with ample substrate scope and broad group tolerance.

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Citations

Jul 14, 2016·The Journal of Organic Chemistry·Aniket MishraIndubhusan Deb
May 4, 2017·The Journal of Organic Chemistry·Shao-Bo WangShu-Li You
Mar 27, 2018·Chemistry, an Asian Journal·Lucien D Caspers, Boris J Nachtsheim
Jul 24, 2018·Chemical Society Reviews·Carlo SambiagioMichael Schnürch
May 5, 2018·Organic & Biomolecular Chemistry·Changduo PanJin-Tao Yu
Mar 17, 2021·Organic & Biomolecular Chemistry·Yu Ru-JianXue-Min Duan
May 31, 2017·Organic Letters·Ruhuai MeiLutz Ackermann
Apr 5, 2018·The Journal of Organic Chemistry·Taejoo JeongIn Su Kim
Jan 29, 2019·The Journal of Organic Chemistry·Rajendra S RohokaleChepuri V Ramana
Oct 27, 2017·The Journal of Organic Chemistry·Aniket MishraIndubhusan Deb
Jan 29, 2022·Organic & Biomolecular Chemistry·Shruti RajputNidhi Jain

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