PMID: 4202581DOI: 10.1016/0006-2952(73)90196-2Dec 1, 1973

Relationship between the inhibition constant (K1) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction

Biochemical Pharmacology
Y Cheng, W H Prusoff

Abstract

No abstract listed.

References

The kinetics of enzyme-catalyzed reactions with two or more substrates or products. I. Nomenclature and rate equations

Jan 8, 1963·Biochimica Et Biophysica Acta·W W CLELAND

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3H-(-)DO 710 discriminates guanine nucleotide sensitive and insensitive dopamine binding sites

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In kitten ventricular myocardium, the inotropic potency of an agonist is determined by both its intrinsic activity for the adenylyl cyclase and its affinity for the beta-adrenoceptors

Aug 1, 1981·Naunyn-Schmiedeberg's Archives of Pharmacology·A J Kaumann

3H-(-)-Bupranolol, a new beta-adrenoceptor radioligand: characterization of its binding to kitten heart beta-adrenoceptors

Aug 1, 1981·Naunyn-Schmiedeberg's Archives of Pharmacology·T H MorrisA J Kaumann

A study of the sensitivity of rat brain alpha 2-adrenoceptors during chronic antidepressant treatments

Aug 1, 1982·Naunyn-Schmiedeberg's Archives of Pharmacology·M F Sugrue

L-654,284 a new potent and selective alpha 2-adrenoceptor antagonist

Jun 1, 1986·Naunyn-Schmiedeberg's Archives of Pharmacology·D J PettiboneJ J Baldwin

Sodium regulation of agonist and antagonist binding to beta-adrenoceptors in intact and Ns-deficient membranes

Jun 1, 1986·Naunyn-Schmiedeberg's Archives of Pharmacology·M Minuth, K H Jakobs

On spare beta-adrenoceptors of inotropic effect of catecholamines in kitten ventricle

Nov 1, 1978·Naunyn-Schmiedeberg's Archives of Pharmacology·A J Kaumann

Interactions of MEN 935 (adimolol), a long acting beta- and alpha-adrenolytic antihypertensive agent, with postsynaptic alpha-adrenoceptors in different isolated blood vessels--influence of angiotensin II

Jul 1, 1986·Naunyn-Schmiedeberg's Archives of Pharmacology·R PallukW D Bechtel

Lesioning of serotoninergic and noradrenergic nerve fibres of the rat brain does not decrease binding of 3H-clonidine and 3H-rauwolscine to cortical membranes

Jan 1, 1985·Naunyn-Schmiedeberg's Archives of Pharmacology·G GrossH J Schümann

Competitive and non-competitive interactions between specific ligands and beta-adrenoceptors in living cardiac cells

Nov 1, 1982·Naunyn-Schmiedeberg's Archives of Pharmacology·H PorzigH Reuter

Differential effects of nifedipine, verapamil, and diltiazem on noradrenaline-induced contractions, adrenergic transmitter release, and alpha-adrenoceptor binding in the female rabbit urethra

May 1, 1984·Naunyn-Schmiedeberg's Archives of Pharmacology·B LarssonK E Andersson

Solubilization and characterization of the 3H-desipramine binding site of rat phaeochromocytoma cells (PC12-cells)

Dec 1, 1986·Naunyn-Schmiedeberg's Archives of Pharmacology·E Schömig, Heinz Bönisch

3H]-Spiroperidol labels dopamine receptors in membranes from rabbit mesenteric artery

Apr 1, 1980·Naunyn-Schmiedeberg's Archives of Pharmacology·O E Brodde, G Gross

Different binding and degradation of proinsulin, insulin and insulin-like growth factor-1 (IGF-1) in cultured renal proximal tubular cells. Implications for the prolonged serum half-life of proinsulin

Jul 1, 1996·Acta Diabetologica·P M JehleF Keller

Beta 1- and beta 2-adrenoceptor binding and functional response in right and left atria of rat heart

Sep 1, 1985·Naunyn-Schmiedeberg's Archives of Pharmacology·E N JubergP W Abel

Xanthine derivatives as antagonists at A1 and A2 adenosine receptors

Sep 1, 1985·Naunyn-Schmiedeberg's Archives of Pharmacology·U SchwabeM J Lohse

Muscarinic acetylcholine receptors in the heart of rats before and after birth

Jan 1, 1986·Pflügers Archiv : European journal of physiology·J NedomaS Tucek

Properties of agonist binding at the beta-adrenoceptor of the rat reticulocyte

Oct 1, 1982·Naunyn-Schmiedeberg's Archives of Pharmacology·G WiemerD Brockmeier

125I] N6-p-Hydroxyphenylisopropyladenosine, a new ligand for Ri adenosine receptors

Oct 1, 1982·Naunyn-Schmiedeberg's Archives of Pharmacology·U SchwabeH Glossmann

No evidence for temperature-dependent changes in the pharmacological specificity of beta 1- and beta 2-adrenoceptors in rabbit lung membranes

Feb 1, 1983·Naunyn-Schmiedeberg's Archives of Pharmacology·O E BroddeA Prywarra

Relationship between the cellular accumulation and the cytotoxicity of S12363, a new Vinca alkaloid derivative

Jan 1, 1992·Cancer Chemotherapy and Pharmacology·A PierréG Atassi

Novel pyrrolo[2,3-d]pyrimidine antifolate TNP-351: cytotoxic effect on methotrexate-resistant CCRF-CEM cells and inhibition of transformylases of de novo purine biosynthesis

Jan 1, 1994·Cancer Chemotherapy and Pharmacology·F ItohG P Beardsley

Identification and characterization of the beta-adrenergic receptor on neuroblastoma x glioma hybrid NG108-15 cells

Sep 1, 1990·Cellular and Molecular Neurobiology·A Ghahary, K W Cheng

Dopamine D1 receptors labelled with [3H]SCH23390 in rabbit cerebral cortex and neostriatum. Equilibrium binding, kinetics and selectivity

Dec 1, 1989·Naunyn-Schmiedeberg's Archives of Pharmacology·T A ReaderK M Dewar

Versatile synthesis of bi- and tri-antennary galactose ligands: interaction with the Gal/GalNAc receptor of human hepatoma cells

Jun 1, 1995·Glycoconjugate Journal·A Kichler, F Schuber

Steroid hormone specifically binds to rat kidney plasma membrane

Dec 1, 1991·Journal of Bioenergetics and Biomembranes·I IbarrolaM Trueba

Prerequisite for His(4) in deltorphin A for highδ opioid receptor selectivity

Oct 1, 1994·Amino Acids·S SalvadoriL H Lazarus

Analysis of 3H-kainic acid binding to brain membranes in rats and frogs

May 1, 1985·Biulleten' eksperimental'noĭ biologii i meditsiny·A M Zharkovskiĭ, T A Zharkovskaia

Dopamine receptors in the developing sheep kidney

Jan 1, 1988·Pediatric Nephrology : Journal of the International Pediatric Nephrology Association·R A FelderP A Jose

Signal transduction pathways of muscarinic receptors in circular smooth muscle from the rabbit caecum

Nov 9, 1994·Molecular and Cellular Biochemistry·P CuqJ P Bali

Effects of sodium, lithium, and magnesium on in vitro binding of [3H]SCH23390 in rat neostriatum and cerebral cortex

May 1, 1989·Neurochemical Research·E GottbergT A Reader

Beta-DL-methylene-aspartate, an inhibitor of aspartate aminotransferase, potently inhibits L-glutamate uptake into astrocytes

Jul 1, 1989·Neurochemical Research·A S BenderH S White

Alpha-1 and alpha-2 adrenoceptor binding in cerebral cortex: role of disulfide and sulfhydryl groups

Jan 1, 1986·Neurochemical Research·T A ReaderL Grondin

Analogs of thyrotropin-releasing hormone (TRH): receptor affinities in brains, spinal cords, and pituitaries of different species

Feb 1, 1991·Neurochemical Research·N A SharifR L Whiting

Stereoselective uptake of the GABA-transaminase inhibitors gamma-vinyl GABA and gamma-acetylenic GABA into neurons and astrocytes

Nov 1, 1986·Neurochemical Research·A SchousboeN Seiler

Similarities of adenosine uptake systems in astrocytes and neurons in primary cultures

Nov 1, 1986·Neurochemical Research·A S Bender, L Hertz

5,8-disubstituted indolizidines: a new class of noncompetitive blockers for nicotinic receptor-channels

Nov 1, 1991·Neurochemical Research·J W DalyR S Aronstam

Muscarinic receptor subtypes in bovine adrenal medulla

Dec 1, 1992·Neurochemical Research·J S AguilarM Criado

Reconstitution of solubilized atrial cholinergic muscarinic receptors in liposomes

Jan 1, 1987·Neurochemical Research·J S AguilarE De Robertis

Direct characterization of beta-adrenoceptors in membranes of immature red blood cells from rats

Dec 15, 1978·Blut·G KaiserD Palm

Expression of functional Y1 receptors for neuropeptide Y in human Ewing's sarcoma cell lines

Jan 1, 1992·Journal of Cancer Research and Clinical Oncology·F van ValenH Jürgens

The aortic alpha 1-adrenergic receptor in familial amyloidotic polyneuropathy

Jan 1, 1988·Journal of Neural Transmission·T AzumaH Yoshida

Alpha-1 and alpha-2 adrenoceptor binding in cerebral cortex: competition studies with [3H]prazosin and [3H]idazoxan

Jan 1, 1987·Journal of Neural Transmission·T A ReaderL Grondin

Neurochemical evidence for a neuronal GABAergic system in the rat sympathetic superior cervical ganglion

Jan 1, 1992·Journal of Neural Transmission. General Section·G González BurgosD P Cardinali

The binding of [3H]-5-hydroxytryptamine to homogenates of human brain

Jan 1, 1982·Journal of Neural Transmission·E DehlinB Winblad

The effect of (+)- and (-)-oxaprotiline administered repeatedly on the dopamine system

Jan 1, 1991·Journal of Neural Transmission. General Section·J MajH Sowińska

3H]205-501, a non-catechol dopaminergic agonist, labels selectively and with high affinity dopamine D2 receptors

Jan 1, 1985·Journal of Neural Transmission·A ClosseR Nordmann

Pharmacological properties of EXP 561, a potential antidepressant drug

Jan 1, 1987·Journal of Neural Transmission·J MajG Nowak

Dopamine agonist activity of EMD 23,448

Jan 1, 1985·Journal of Neural Transmission·G E Martin, D J Pettibone

Effects of tranylcypromine enantiomers on monoamine uptake and release and imipramine binding

Jan 1, 1986·Journal of Neural Transmission·J Tuomisto, D F Smith

Autoradiographic localization of dopamine D2-like receptors in the rabbit pulmonary vascular tree

Jun 1, 1994·Naunyn-Schmiedeberg's Archives of Pharmacology·Y KobayashiF Amenta

SDZ PSD 958, a novel D1 receptor antagonist with potential limbic selectivity

Jan 1, 1996·Journal of Neural Transmission·R MarksteinD Hoyer

Atypical in vitro and in vivo binding of [3H]S-14506 to brain 5-HT1A receptors

Jan 1, 1997·Journal of Neural Transmission·L LimaM Hamon

D1 receptor binding in rat striatum: modification by various D1 and D2 antagonists, but not by sibutramine hydrochloride, antidepressants or treatments which enhance central dopaminergic function

Jan 1, 1995·Journal of Neural Transmission. General Section·S C CheethamD J Heal

SDZ GLC 756, a novel octahydrobenzo[g]quinoline derivative exerts opposing effects on dopamine D1 and D2 receptors

Jan 1, 1996·Journal of Neural Transmission·R MarksteinD Hoyer

Muscarinic receptors and amylase secretion of rat pancreatic acini during cerulein-induced acute pancreatitis

Aug 1, 1987·Digestive Diseases and Sciences·J MorissetL Larose

3H] Dihydroergonine binding to alpha-adrenergic receptors in human platelets

Jan 1, 1978·Klinische Wochenschrift·K H Jakobs, R Rauschek

Strategic approaches to drug design. II. Modelling studies on phosphodiesterase substrates and inhibitors

Jul 1, 1987·Journal of Computer-aided Molecular Design·A DavisJ G Vinter

The influence of hydrochlorothiazide on the pharmacokinetics of enalapril in elderly patients

Jan 1, 1992·European Journal of Clinical Pharmacology·K WeisserE Mutschler

Androgens inhibit basal and estrogen-induced cell proliferation in the ZR-75-1 human breast cancer cell line

Oct 1, 1988·Breast Cancer Research and Treatment·R PoulinF Labrie

Antiestrogenic properties of keoxifene, trans-4-hydroxytamoxifen, and ICI 164384, a new steroidal antiestrogen, in ZR-75-1 human breast cancer cells

Oct 1, 1989·Breast Cancer Research and Treatment·R PoulinF Labrie

Multiple actions of synthetic 'progestins' on the growth of ZR-75-1 human breast cancer cells: an in vitro model for the simultaneous assay of androgen, progestin, estrogen, and glucocorticoid agonistic and antagonistic activities of steroids

Jan 1, 1991·Breast Cancer Research and Treatment·R PoulinF Labrie

Androgen and glucocorticoid receptor-mediated inhibition of cell proliferation by medroxyprogesterone acetate in ZR-75-1 human breast cancer cells

Mar 1, 1989·Breast Cancer Research and Treatment·R PoulinF Labrie

The influence of ageing on muscarinic receptors, beta-adrenoceptors and adenylate cyclase activity in the bovine lung

Jan 1, 1995·Veterinary Research Communications·E Roets, C Burvenich

Effects of local anesthetics on phospholipid topology and dopamine uptake and release in rat brain synaptosomes

Jan 1, 1982·The Journal of Membrane Biology·P G Bradford, G V Marinetti

Muscarinic responses of gastric parietal cells

Jun 1, 1991·The Journal of Membrane Biology·J M WilkesG Sachs

Molecular environment of the phencyclidine binding site in the nicotinic acetylcholine receptor membrane

Jun 1, 1991·The Journal of Membrane Biology·A L Palma, H Wang

The carboxy-terminal region of human interleukin-5 is essential for maintenance of tertiary structure but not for dimerization

Jul 1, 1996·Journal of Protein Chemistry·A E ProudfootT N Wells

Desensitization pattern of cardiac beta-adrenoceptor subtypes by prolonged in vivo infusion of pindolol and celiprolol in rats

Jan 1, 1990·Basic Research in Cardiology·C NanoffH Pittner

Binding of [3H]ouabain to endothelial cells derived from various vascular beds

Nov 1, 1987·Basic Research in Cardiology·M FreissmuthW Schütz

Flavonoid compounds are potent inhibitors of cyclic AMP phosphodiesterase

Aug 15, 1978·Experientia·A BeretzJ C Stoclet

3[H]-Sulpiride labels mesolimbic non-dopaminergic sites that bind antidepressant drugs

Nov 15, 1985·Experientia·J G CsernanskyL E Hollister

Hypotensive activity of PAF-acether in rats

Dec 1, 1982·Agents and Actions·C G CaillardL Julou

Specific binding of [3H]mepyramine to histamine H1-receptors in vascular smooth muscle membranes

Apr 1, 1983·Agents and Actions·M Carman-Krzan

Monoamine oxidase inhibition by d-amphetamine in ganglia and nerve endings

Jul 15, 1982·Experientia·E J Filinger, F J Stefano

The effect of group selective reagents N-ethylmaleimide and dithiothreitol on histamine H1-receptor binding sites in the vascular smooth muscle membranes

Apr 1, 1984·Agents and Actions·M Carman-Krzan

The oxime HGG-12 as a muscarinic acetylcholine receptor antagonist without intrinsic activity in cardiac membranes

Jan 1, 1991·Archives of Toxicology·C ReithmannK Werdan

Characterization of vascular histamine H1-receptors: multiple affinity states of aortic histamine H1-receptor

Apr 1, 1985·Agents and Actions·M Carman-Krzan

Effects of pheochromocytoma on cardiovascular alpha adrenergic receptor system

Aug 1, 1985·Heart and Vessels·G TsujimotoB B Hoffman

Computer modelling of the binding of non-selective ligands to biological receptors

Dec 16, 1983·Pharmaceutisch Weekblad. Scientific Edition·H J WynneW Soudijn

Characterization of binding of 3H-SCH 23390 to dopamine D-1 receptors. Correlation to other D-1 and D-2 measures and effect of selective lesions

Jan 1, 1987·Journal of Neural Transmission·J Hyttel, J Arnt

Beta-adrenergic receptors in DMBA-induced rat mammary tumors: correlation with progesterone receptor and tumor growth

Jul 1, 1989·Breast Cancer Research and Treatment·B MarchettiF Labrie

Beta-adrenergic receptor subtypes in iris-ciliary body of rabbits

Jan 1, 1984·Graefe's Archive for Clinical and Experimental Ophthalmology = Albrecht Von Graefes Archiv Für Klinische Und Experimentelle Ophthalmologie·C J SchmittN N Share

A study on the ocular and extraocular pharmacology of metipranolol

Jan 1, 1985·Graefe's Archive for Clinical and Experimental Ophthalmology = Albrecht Von Graefes Archiv Für Klinische Und Experimentelle Ophthalmologie·M F SugrueM P Viader

Histaminergic H1-receptors in smooth muscle and endothelium of bovine thoracic aorta

Apr 1, 1989·Agents and Actions·M Carman-Krzan

Choroid plexus epithelial cells in primary culture: a model of 5HT1C receptor activation by hallucinogenic drugs

Jan 1, 1991·Psychopharmacology·E Sanders-Bush, M Breeding

Electrophysiological, biochemical and behavioral evidence for 5-HT2 and 5-HT3 mediated control of dopaminergic function

Jan 1, 1993·Psychopharmacology·M G PalfreymanA A Carr

Etoperidone, trazodone and MCPP: in vitro and in vivo identification of serotonin 5-HT1A (antagonistic) activity

Jan 1, 1992·Psychopharmacology·R B RaffaJ L Vaught

The pharmacology of VA21B7: an atypical 5-HT3 receptor antagonist with anxiolytic-like properties in animal models

Jan 1, 1995·Psychopharmacology·Inés ArtaizJ Del Río

Novel alkoxy-oxazolyl-tetrahydropyridine muscarinic cholinergic receptor antagonists

Jan 1, 1995·Psychopharmacology·H E ShannonC H Mitch

Repeated ketamine administration produces up-regulation of muscarinic acetylcholine receptors in the forebrain, and reduces behavioral sensitivity to scopolamine in mice

Feb 1, 1995·Psychopharmacology·T MoritaH Kuribara

BRL 46470A: a highly potent, selective and long acting 5-HT3 receptor antagonist with anxiolytic-like properties

Jan 1, 1993·Psychopharmacology·T BlackburnM D Wood

Endogenous dopamine limits the binding of antipsychotic drugs to D3 receptors in the rat brain: a quantitative autoradiographic study

Nov 1, 1996·The Histochemical Journal·A SchotteJ E Leysen

Concerning the way to study the relative potencies of bronchodilator agents in vitro

Jan 1, 1986·Lung·J A Raaijmakers, R J van Rozen

Comparative biochemical pharmacology of central nervous system dopamine D1 and D2 receptors

Jan 1, 1992·Molecular Neurobiology·T A ReaderK M Dewar

Comparison of R-, S-, and RS-albuterol interaction with human beta 1- and beta 2-adrenergic receptors

Jan 1, 1996·Clinical Reviews in Allergy & Immunology·R B PennJ L Benovic

Protein engineering of de novo protein with predesigned structure and activity

Oct 1, 1996·Applied Biochemistry and Biotechnology·D A DolgikhM P Kirpichnikov

Inhibition of thymidylate synthase by the diastereoisomers of leucovorin

Jan 1, 1990·Cancer Chemotherapy and Pharmacology·P P Lee, R L Schilsky

The next frontier in the molecular biology of the opioid system. The opioid receptors

Jan 1, 1987·Molecular Neurobiology·O CivelliD Grandy

Pharmacological characterization of (10bS)-1,2,3,5,6,10b-hexahydropyrrolo[2,1-a]isoquinoline oxalate (YSL-3S) as a new alpha2-adrenoceptor antagonist

Sep 8, 2000·Archives of Pharmacal Research·S H ChungC Jin

Pharmacological characterization of LB50016, N-(4-amino)butyl 3-phenylpyrrolidine derivative, as a new 5-HT1A receptor agonist

May 7, 1999·Archives of Pharmacal Research·C H LeeY Z Kim

Selectivity of oxomemazine for the M1 muscarinic receptors

Dec 1, 1994·Archives of Pharmacal Research·S W LeeJ G Kim

Evaluation of radioiodinated 5-iodo-3-(2(S)-azetidinylmethoxy)pyridine as a ligand for SPECT investigations of brain nicotinic acetylcholine receptors

Jul 20, 2002·Annals of Nuclear Medicine·Hideo SajiTakahiro Mukai

Effect of encainide, ODE, MODE, and flecainide on ADP/5-HT induced platelet aggregation and in the anesthetized dog coronary artery stenosis-occlusion model of intravascular thrombosis

Aug 1, 1991·Cardiovascular Drugs and Therapy·J S FlemingM J Antonaccio

Attenuation of muscarinic receptor-G-protein interaction in Alzheimer disease

Jan 1, 1995·Molecular and Chemical Neuropathology·G Ferrari-DiLeoD D Flynn

Inhibition of platelet aggregation by adenosine receptor agonists

Jun 1, 1994·Naunyn-Schmiedeberg's Archives of Pharmacology·Gloria CristalliR A Olsson

The diterpenoid alkaloid noroxoaconitine is a Mapkap kinase 5 (MK5/PRAK) inhibitor

Jul 20, 2010·Cellular and Molecular Life Sciences : CMLS·Sergiy KostenkoUgo Moens

Serotonin transporter activity of imidazolidine-2,4-dione and imidazo[2,1-f]purine-2,4-dione derivatives in aspect of their acid-base properties

Oct 11, 2012·Medicinal Chemistry Research : an International Journal for Rapid Communications on Design and Mechanisms of Action of Biologically Active Agents·Agnieszka ZagórskaGabriel Nowak

Selectivity of repaglinide and glibenclamide for the pancreatic over the cardiovascular K(ATP) channels

Jul 26, 2006·Diabetologia·Damian StephanUlrich Quast

Fluorescence study on site-specific binding of perfluoroalkyl acids to human serum albumin

Oct 16, 2008·Archives of Toxicology·Yan-Min Chen, Liang-Hong Guo

3H]LY334370, a novel radioligand for the 5-HT1F receptor. I. In vitro characterization of binding properties

May 19, 2005·Naunyn-Schmiedeberg's Archives of Pharmacology·D B WainscottD L Nelson

The novel suramin analogue NF864 selectively blocks P2X1 receptors in human platelets with potency in the low nanomolar range

Sep 15, 2005·Naunyn-Schmiedeberg's Archives of Pharmacology·Susanne HornerG Lambrecht

Agonist effects of zinterol at the mouse and human beta(3)-adrenoceptor

Apr 8, 2006·Naunyn-Schmiedeberg's Archives of Pharmacology·Dana S HutchinsonTore Bengtsson

Cell and tissue responses of a range of Urotensin II analogs at cloned and native urotensin II receptors. Evidence for coupling promiscuity

Apr 6, 2006·Naunyn-Schmiedeberg's Archives of Pharmacology·Wei SongD G Lambert

Comparison of three radioligands for the labelling of human beta-adrenoceptor subtypes

Oct 10, 2006·Naunyn-Schmiedeberg's Archives of Pharmacology·Nadja NiclaussMartin C Michel

Striking differences of action of lisuride stereoisomers at histamine H1 receptors

Nov 16, 2006·Naunyn-Schmiedeberg's Archives of Pharmacology·Heinz H PertzAndrea Strasser

The in vitro pharmacology of the peripherally restricted opioid receptor antagonists, alvimopan, ADL 08-0011 and methylnaltrexone

Mar 7, 2007·Naunyn-Schmiedeberg's Archives of Pharmacology·David T BeattieR Vickery

In vitro pharmacological characterisation of a novel cyclic nociceptin/orphanin FQ analogue c[Cys(7,10)]N/OFQ(1-13)NH (2)

Jun 29, 2007·Naunyn-Schmiedeberg's Archives of Pharmacology·Masato KitayamaD G Lambert

Molecular cloning and functional expression of the murine noradrenaline transporter

Sep 21, 2007·Naunyn-Schmiedeberg's Archives of Pharmacology·Andrea MuckHeinz Bönisch

The in vitro pharmacological profile of TD-5108, a selective 5-HT(4) receptor agonist with high intrinsic activity

Apr 17, 2008·Naunyn-Schmiedeberg's Archives of Pharmacology·J A M SmithP P A Humphrey

In vitro and in vivo pharmacological analysis of imidazole-free histamine H3 receptor antagonists: promising results for a brain-penetrating H3 blocker with weak anticholinesterase activity

May 23, 2008·Naunyn-Schmiedeberg's Archives of Pharmacology·Simona BertoniElisabetta Barocelli

Subnanomolar dopamine D3 receptor antagonism coupled to moderate D2 affinity results in favourable antipsychotic-like activity in rodent models: I. neurochemical characterisation of RG-15

Jun 14, 2008·Naunyn-Schmiedeberg's Archives of Pharmacology·Béla KissZsolt Szombathelyi

Functional reconstitution of the human chemokine receptor CXCR4 with G(i)/G (o)-proteins in Sf9 insect cells

Jun 5, 2008·Naunyn-Schmiedeberg's Archives of Pharmacology·Patrick KleemannRoland Seifert

Binding of the novel radioligand [(3)H]UFP-101 to recombinant human and native rat nociceptin/orphanin FQ receptors

Sep 23, 2008·Naunyn-Schmiedeberg's Archives of Pharmacology·Massimo IbbaD G Lambert

Interaction of the human plasma membrane monoamine transporter (hPMAT) with antidepressants and antipsychotics

Dec 17, 2009·Naunyn-Schmiedeberg's Archives of Pharmacology·Britta Haenisch, Heinz Bönisch

Inhibition of monoamine oxidase activity by cannabinoids.

Apr 20, 2010·Naunyn-Schmiedeberg's Archives of Pharmacology·Zdenek Fisar

Establishment of recombinant cannabinoid receptor assays and characterization of several natural and synthetic ligands

Jul 10, 2010·Naunyn-Schmiedeberg's Archives of Pharmacology·Sarah GeigerJörg Heilmann

N (α)-Methylated phenylhistamines exhibit affinity to the hH(4)R-a pharmacological and molecular modelling study

Jul 30, 2011·Naunyn-Schmiedeberg's Archives of Pharmacology·Hans-Joachim WittmannAndrea Straber

Role of the second and third extracellular loops of the histamine H(4) receptor in receptor activation

Jul 30, 2011·Naunyn-Schmiedeberg's Archives of Pharmacology·Irena BrunskoleArmin Buschauer

δ-Aminolevulinic acid and its methyl ester induce the formation of Protoporphyrin IX in cultured sensory neurones

Sep 29, 2011·Naunyn-Schmiedeberg's Archives of Pharmacology·B NovakH Lübbert

Characterization of a novel, brain-penetrating CB1 receptor inverse agonist: metabolic profile in diet-induced obese models and aspects of central activity

Sep 29, 2011·Naunyn-Schmiedeberg's Archives of Pharmacology·Laura H JacobsonSandra Teixeira

Interactions of recombinant human histamine H₁R, H₂R, H₃R, and H₄R receptors with 34 antidepressants and antipsychotics

Oct 29, 2011·Naunyn-Schmiedeberg's Archives of Pharmacology·Heidrun ApplRoland Seifert

Role of the amino-terminal transmembrane domain of sulfonylurea receptor SUR2B for coupling to K(IR)6.2, ligand binding, and oligomerization

Nov 18, 2011·Naunyn-Schmiedeberg's Archives of Pharmacology·Marcus WinklerUlrich Quast

Importance of the Kir6.2 N-terminus for the interaction of glibenclamide and repaglinide with the pancreatic K(ATP) channel

Nov 16, 2011·Naunyn-Schmiedeberg's Archives of Pharmacology·Petra KühnerUlrich Quast

Interaction of antidepressant and antipsychotic drugs with the human organic cation transporters hOCT1, hOCT2 and hOCT3

Jul 19, 2012·Naunyn-Schmiedeberg's Archives of Pharmacology·Britta HaenischHeinz Bönisch

The in vitro pharmacological profile of TD-1211, a neutral opioid receptor antagonist

Apr 4, 2013·Naunyn-Schmiedeberg's Archives of Pharmacology·Pamela R TsurudaDavid T Beattie

Extracellular loop 3 of the noradrenaline transporter contributes to substrate and inhibitor selectivity

Oct 2, 2013·Naunyn-Schmiedeberg's Archives of Pharmacology·Timothy LynaghLesley J Bryan-Lluka

Pharmacological profile of astemizole-derived compounds at the histamine H1 and H4 receptor--H1/H4 receptor selectivity

Nov 19, 2013·Naunyn-Schmiedeberg's Archives of Pharmacology·Eva WagnerAndrea Strasser

Pharmacological characterization of N1-(2-methoxyphenyl)-N4-hexylpiperazine as a multi-target antagonist of α1A/α1D-adrenoceptors and 5-HT1A receptors that blocks prostate contraction and cell growth

Nov 12, 2013·Naunyn-Schmiedeberg's Archives of Pharmacology·Fernanda Chagas-SilvaClaudia Lucia Martins Silva

Metabotropic glutamate 2 receptor potentiators: receptor modulation, frequency-dependent synaptic activity, and efficacy in preclinical anxiety and psychosis model(s)

Feb 18, 2005·Psychopharmacology·Michael P JohnsonDarryle D Schoepp

Preclinical pharmacology of F-98214-TA, a novel potent serotonin and norepinephrine uptake inhibitor with antidepressant and anxiolytic properties

Jul 21, 2005·Psychopharmacology·Inés ArtaizAurelio Orjales

MDMA (Ecstasy) and human dopamine, norepinephrine, and serotonin transporters: implications for MDMA-induced neurotoxicity and treatment

Oct 13, 2005·Psychopharmacology·Christopher D VerricoBertha K Madras

In vitro and in vivo studies in rats with LY293558 suggest AMPA/kainate receptor blockade as a novel potential mechanism for the therapeutic treatment of anxiety disorders

Feb 14, 2006·Psychopharmacology·Andrew AltJeffrey M Witkin

WAY-100635 is a potent dopamine D4 receptor agonist

Aug 18, 2006·Psychopharmacology·Benjamin R ChemelDavid E Nichols

Ligands selective for alpha4beta2 but not alpha3beta4 or alpha7 nicotinic receptors generalise to the nicotine discriminative stimulus in the rat

Nov 23, 2006·Psychopharmacology·Janice W SmithMark Tricklebank

Interaction of the novel antipsychotic aripiprazole with 5-HT1A and 5-HT 2A receptors: functional receptor-binding and in vivo electrophysiological studies

Jan 24, 2007·Psychopharmacology·Arlene D StarkKevin D Burris

Pharmacology of neuropeptide S in mice: therapeutic relevance to anxiety disorders

Mar 4, 2008·Psychopharmacology·Sarah K LeonardRobert H Ring

Dopamine D4 receptor involvement in the discriminative stimulus effects in rats of LSD, but not the phenethylamine hallucinogen DOI

Jul 8, 2008·Psychopharmacology·Danuta Marona-LewickaDavid E Nichols

RO4938581, a novel cognitive enhancer acting at GABAA alpha5 subunit-containing receptors

Oct 22, 2008·Psychopharmacology·Theresa M BallardMaria-Clemencia Hernandez

Kappa opioid mediation of cannabinoid effects of the potent hallucinogen, salvinorin A, in rodents

Apr 1, 2010·Psychopharmacology·D Matthew WalentinyJenny L Wiley

Clozapine and other competitive antagonists reactivate risperidone-inactivated h5-HT7 receptors: radioligand binding and functional evidence for GPCR homodimer protomer interactions

Sep 10, 2010·Psychopharmacology·Milt TeitlerCarol Smith

Pharmacological and behavioral characterization of the 5-HT2A receptor in C57BL/6N mice

Feb 23, 2011·Psychopharmacology·John P Dougherty, Vincent J Aloyo

Inhibitory potencies of trimipramine and its main metabolites at human monoamine and organic cation transporters

Apr 13, 2011·Psychopharmacology·Britta HaenischHeinz Bönisch

Involvement of histamine receptors in the atypical antipsychotic profile of clozapine: a reassessment in vitro and in vivo

Sep 14, 2011·Psychopharmacology·Marie Humbert-ClaudeJean-Michel Arrang

Substituted heteroaromatic compounds: effect on nicotine self-administration in rats

Jan 6, 2012·Psychopharmacology·John R CashmanMarc R Azar

Relations between stimulation of mesolimbic dopamine and place conditioning in rats produced by cocaine or drugs that are tolerant to dopamine transporter conformational change

Apr 25, 2013·Psychopharmacology·Gianluigi TandaJonathan L Katz

Behavioral and neurochemical pharmacology of six psychoactive substituted phenethylamines: mouse locomotion, rat drug discrimination and in vitro receptor and transporter binding and function

Oct 22, 2013·Psychopharmacology·Amy J EshlemanMichael B Gatch

Determination of drug-serum protein interactions via fluorescence polarization measurements

Jun 8, 2007·Analytical and Bioanalytical Chemistry·Ulf Mathias, Manfred Jung

Expanding the scope of MS binding assays to low-affinity markers as exemplified for mGAT1

Mar 18, 2008·Analytical and Bioanalytical Chemistry·Christine ZepperitzKlaus T Wanner

Ligand-binding assays for cyanobacterial neurotoxins targeting cholinergic receptors

Mar 20, 2010·Analytical and Bioanalytical Chemistry·Rómulo AráozJordi Molgó

Beta-secretase as a target for Alzheimer's disease drug discovery: an overview of in vitro methods for characterization of inhibitors

Apr 20, 2011·Analytical and Bioanalytical Chemistry·Francesca ManciniVincenza Andrisano

Detection of flagellin by interaction with human recombinant TLR5 immobilized in liposomes

Nov 28, 2012·Analytical and Bioanalytical Chemistry·Y OlguínR Galindo

Fluorescent system based on bacterial expression of hybrid KcsA channels designed for Kv1.3 ligand screening and study

Jan 12, 2013·Analytical and Bioanalytical Chemistry·Kseniya S KudryashovaAlexey V Feofanov

Towards metabolically stable 5-HT7 receptor ligands: a study on 1-arylpiperazine derivatives and related isosters

Apr 11, 2013·Experimental Brain Research·Enza LacivitaMarcello Leopoldo

Multiple conformations of 5-HT2A and 5-HT 2C receptors in rat brain: an autoradiographic study with [125I](±)DOI

Jul 19, 2013·Experimental Brain Research·Juan F López-GiménezGuadalupe Mengod

Modeling of cellular arginine uptake by more than one transporter

Nov 25, 2011·The Journal of Membrane Biology·Marietha J NelGeoffrey P Candy

The most common Chinese rhesus macaque MHC class I molecule shares peptide binding repertoire with the HLA-B7 supertype

May 19, 2010·Immunogenetics·Christopher SolomonBianca R Mothé

Functional analysis of frequently expressed Chinese rhesus macaque MHC class I molecules Mamu-A1*02601 and Mamu-B*08301 reveals HLA-A2 and HLA-A3 supertypic specificities

Jan 29, 2011·Immunogenetics·Scott SouthwoodAlessandro Sette

The role of MHC class I allele Mamu-A*07 during SIV(mac)239 infection

Jul 7, 2011·Immunogenetics·Jason S ReedNancy A Wilson

Synthesis and evaluation of radioiodinated (S,S)-2-(alpha-(2-iodophenoxy)benzyl)morpholine for imaging brain norepinephrine transporter

Mar 9, 2006·European Journal of Nuclear Medicine and Molecular Imaging·Naoki KanegawaHideo Saji

Reversibility of ecstasy-induced reduction in serotonin transporter availability in polydrug ecstasy users

Sep 1, 2005·European Journal of Nuclear Medicine and Molecular Imaging·Ralph BuchertMalte Clausen

Molecular imaging of alpha7 nicotinic acetylcholine receptors: design and evaluation of the potent radioligand [18F]NS10743

Jan 13, 2009·European Journal of Nuclear Medicine and Molecular Imaging·Winnie Deuther-ConradPeter Brust

Human breast cell lines exhibit functional alpha2-adrenoceptors

Nov 18, 2005·Cancer Chemotherapy and Pharmacology·Stella Maris VázquezIsabel Alicia Lüthy

hPEPT1 is responsible for uptake and transport of Gly-Sar in the human bronchial airway epithelial cell-line Calu-3

Dec 21, 2007·Pflügers Archiv : European journal of physiology·Helle Bach SøndergaardCarsten Uhd Nielsen

The interconversion of ACC deaminase and D-cysteine desulfhydrase by directed mutagenesis

Oct 1, 2008·Planta·Biljana Todorovic, Bernard R Glick

The antinociceptive effect of intrathecal tramadol in rats: the role of alpha 2-adrenoceptors in the spinal cord

Nov 1, 2011·Journal of Anesthesia·Cai LiKe-Xuan Liu

Dimethyltryptamine and other hallucinogenic tryptamines exhibit substrate behavior at the serotonin uptake transporter and the vesicle monoamine transporter

Sep 17, 2009·Journal of Neural Transmission·Nicholas V CozziArnold E Ruoho

An improved approach to steady-state analysis of monoamine oxidases

Jun 7, 2011·Journal of Neural Transmission·Rona R RamsayAndrew Holt

In vivo biosynthesis of an Ala-scan library based on the cyclic peptide SFTI-1

Aug 18, 2009·Amino Acids·Jeffrey AustinJulio A Camarero

A novel halogen bond and a better-known hydrogen bond cooperation of neonicotinoid and insect nicotinic acetylcholine receptor recognition

Mar 20, 2012·Journal of Molecular Modeling·Hongxia DuanShuhui Jin

Redefining XynA from Penicillium funiculosum IMI 378536 as a GH7 cellobiohydrolase

Jul 11, 2012·Journal of Industrial Microbiology & Biotechnology·Hélène TexierMichael J O'Donohue

Affinity labeling mu opioid receptors with novel radioligands

Aug 3, 2005·Cellular and Molecular Neurobiology·Ke YangG W Pasternak

Creatine and antioxidant treatment prevent the inhibition of creatine kinase activity and the morphological alterations of C6 glioma cells induced by the branched-chain alpha-keto acids accumulating in maple syrup urine disease

Apr 25, 2006·Cellular and Molecular Neurobiology·Cláudia FunchalMoacir Wajner

Kinetics and pharmacology of the D1- and D2-like dopamine receptors in Japanese quail brain

Mar 31, 2009·Cellular and Molecular Neurobiology·Lubica KubíkováLubor Kostál

Decreased GABAA receptors functional regulation in the cerebral cortex and brainstem of hypoxic neonatal rats: effect of glucose and oxygen supplementation

Dec 25, 2009·Cellular and Molecular Neurobiology·T R AnjuC S Paulose

The PG500 series: novel heparan sulfate mimetics as potent angiogenesis and heparanase inhibitors for cancer therapy

Apr 10, 2009·Investigational New Drugs·K DredgeI Bytheway

In vitro antitumor mechanism of a novel cyclin-dependent kinase inhibitor CDKI-83

Feb 19, 2011·Investigational New Drugs·Xiangrui LiuShudong Wang

QSAR analyses on avian influenza virus neuraminidase inhibitors using CoMFA, CoMSIA, and HQSAR

Nov 15, 2006·Journal of Computer-aided Molecular Design·Mingyue ZhengHualiang Jiang

Generation of a homology model of the human histamine H(3) receptor for ligand docking and pharmacophore-based screening

Aug 2, 2007·Journal of Computer-aided Molecular Design·Birgit SchlegelWolfgang Sippl

Fragment-based lead generation: identification of seed fragments by a highly efficient fragment screening technology

Jun 18, 2009·Journal of Computer-aided Molecular Design·Lars NeumannDoris Hafenbradl

Prediction of protein-ligand binding affinity by free energy simulations: assumptions, pitfalls and expectations

May 29, 2010·Journal of Computer-aided Molecular Design·Julien Michel, Jonathan W Essex

Interaction of clozapine and its nitrenium ion with rat D2 dopamine receptors: in vitro binding and computational study

Dec 25, 2010·Journal of Computer-aided Molecular Design·Sébastien Dilly, Jean-François Liégeois

Free enthalpies of replacing water molecules in protein binding pockets

Dec 19, 2012·Journal of Computer-aided Molecular Design·Sereina RinikerWilfred F van Gunsteren

Investigating the hydrogen-bond acceptor site of the nicotinic pharmacophore model: a computational and experimental study using epibatidine-related molecular probes

Nov 28, 2013·Journal of Computer-aided Molecular Design·Clelia DallanoceMarco De Amici

Binding properties of water-soluble carbosilane dendrimers

Sep 2, 2008·Journal of Fluorescence·Elzbieta PedziwiatrMa Angeles Muñoz-Fernandez

An integrated pharmacokinetic-pharmacodynamic model for an Aurora kinase inhibitor

Aug 10, 2010·Journal of Pharmacokinetics and Pharmacodynamics·Hiroko KameiFordyce A Davidson

Segment-dependent expression of muscarinic acetylcholine receptors and G-protein coupling in the equine respiratory tract

Dec 21, 2006·Veterinary Research Communications·G AbrahamF R Ungemach

2- and 8-alkynyl-9-ethyladenines: Synthesis and biological activity at human and rat adenosine receptors

Apr 12, 2008·Purinergic Signalling·Rosaria VolpiniGloria Cristalli

Pyrazolo-triazolo-pyrimidines as adenosine receptor antagonists: Effect of the N-5 bond type on the affinity and selectivity at the four adenosine receptor subtypes

Mar 28, 2008·Purinergic Signalling·Chiara BolcatoStefano Moro

Synthesis and pharmacological characterization of [(125)I]MRS1898, a high-affinity, selective radioligand for the rat A(3) adenosine receptor

Jun 6, 2008·Purinergic Signalling·Zhan-Guo GaoK A Jacobson

Study on the binding interaction between perfluoroalkyl acids and DNA

May 7, 2013·Environmental Science and Pollution Research International·Jie CaoLiang-Hong Guo

Predictions of enzymatic parameters: a mini-review with focus on enzymes for biofuel

Jul 3, 2013·Applied Biochemistry and Biotechnology·Shaomin Yan, Guang Wu

A selective androgen receptor modulator with minimal prostate hypertrophic activity enhances lean body mass in male rats and stimulates sexual behavior in female rats

Nov 10, 2007·Endocrine·George F AllanScott G Lundeen

Design and implementation of high throughput screening assays

Sep 25, 2010·Molecular Biotechnology·Ricardo Macarrón, Robert P Hertzberg

Measuring and interpreting the selectivity of protein kinase inhibitors

Jul 2, 2009·Journal of Chemical Biology·Lynette A Smyth, Ian Collins

Characteristics of an adenosine A1 binding site in human placental membranes

Jan 1, 1989·Archives of Biochemistry and Biophysics·C WorkI H Fox

Human deoxycytidine kinase. Purification and characterization of the cytoplasmic and mitochondrial isozymes derived from blast cells of acute myelocytic leukemia patients

Apr 12, 1977·Biochimica Et Biophysica Acta·Y ChengL S Lee

Discrimination between subclasses of human high-density lipoproteins by the HDL binding sites of bovine liver

Jan 3, 1986·Biochimica Et Biophysica Acta·C M MendelJ P Kane

Properties of herpes simplex virus type 1 and type 2 DNA polymerase

Sep 19, 1980·Biochimica Et Biophysica Acta·M Ostrander, Y Cheng

Interactions between adenylate cyclase inhibitors and beta-adrenoceptors in isolated human fat cells

Jun 15, 1989·Biochemical and Biophysical Research Communications·F Lönnqvist, P Arner

Structure-binding-activity analysis of beta-adrenergic amines--I. Binding to the beta receptor and activation of adenylate cyclase

May 15, 1978·Biochemical Pharmacology·J P BilezikianD E Gammon

Beta-adrenergic receptors and adenylate cyclase activity in rat reticulocytes and mature erythrocytes

Jan 1, 1979·Biochemical Pharmacology·B S Beckman, M D Hollenberg

The effect of lipophilic compounds upon the activity of rat liver mitochondrial monoamine oxidase-A and -B

Apr 15, 1980·Biochemical Pharmacology·C J FowlerK F Tipton

Presence of histamine and serotonin receptors associated with adenylate cyclase in cultured calf-aorta smooth muscle cells. Pharmacological characterization of the histamine response

Dec 1, 1980·Biochemical Pharmacology·A R Luchins, M H Makman

Effects of fluoro-dopamines on dopamine receptors (D1, D2, D3, sites)

Nov 1, 1981·Biochemical Pharmacology·G FirnauK L Kirk

Identification and chemical characterisation of beta-adrenergic receptors in intact turkey erythrocytes

Oct 1, 1981·Biochemical Pharmacology·C AndréA D Strosberg

On the binding of a 3-alpha-methylated digitoxigenin-glucoside to ouabain receptors in heart muscle homogenate

Aug 1, 1982·Biochemical Pharmacology·H Lüllmann, K Mohr

Effects of full and partial beta-adrenergic agonists and antagonists on human lung adenylate cyclase

Jun 15, 1983·Biochemical Pharmacology·M DelhayeJ Christophe

Identification and characterization of alpha 1-adrenergic receptors in human myometrium by [3H]prazosin binding

Mar 1, 1983·Biochemical Pharmacology·S BottariA Vokaer

Alpha-adrenergic potentiation of beta-adrenergic stimulation of rat pineal N-acetyltransferase. Studies using cirazoline and fluorine analogs of norepinephrine

Dec 15, 1984·Biochemical Pharmacology·D SugdenC R Creveling

Thermodynamics of the interactions of tricyclic drugs with binding sites for [3H]imipramine in mouse cerebral cortex

Dec 15, 1984·Biochemical Pharmacology·M E ReithA Lajtha

Desensitization of beta-adrenergic receptor-coupled adenylate cyclase activity. Differences following exposure of cells to two full agonists

Nov 15, 1984·Biochemical Pharmacology·R N PittmanP B Molinoff

Effects of idazoxan on catecholamine systems in rat brain

Aug 15, 1984·Biochemical Pharmacology·D S WalterP W Dettmar

Beta-adrenergic activity and conformation of the antihypertensive specific alpha 2-agonist drug, guanabenz

Feb 15, 1985·Biochemical Pharmacology·S DiamantD Atlas

Identification and characterization of leukotriene D4 receptors in adult and fetal human lung

Dec 15, 1985·Biochemical Pharmacology·M A LewisS T Crooke

Binding characteristics of the dopamine uptake inhibitor [3H]nomifensine to striatal membranes

Apr 15, 1985·Biochemical Pharmacology·M L Dubocovich, N R Zahniser

Heterogeneity between soluble human and rabbit splenic alpha 2-adrenoceptors

Oct 15, 1986·Biochemical Pharmacology·R M McKernanP S Sever

A water-soluble derivative of prazosin prazosinamine hydrochloride [1-(4'-amino-6',7'-dimethoxyquinazolin-2'-yl)-4-(6''-aminohexanoyl) piperazine hydrochloride], reversibly inhibits the calcium-mobilizing action of alpha 1-adrenergic agonists in the perfused rat liver

May 15, 1987·Biochemical Pharmacology·W L ArmaregoF L Bygrave

In vitro pharmacologic activity of congener derivatives and model conjugates of propranolol and practolol

Jul 1, 1987·Biochemical Pharmacology·M M KhanK L Melmon

Characterization of histamine type 1 receptors on natural suppressor lymphoid cells

Nov 15, 1987·Biochemical Pharmacology·M M KhanK L Melmon

Calcium channels in normal and dystrophic hamster cardiac muscle. [3H]nitrendipine binding studies

Aug 15, 1987·Biochemical Pharmacology·S E Howlett, T Gordon

Effect of daunorubicin on dihydropyridine-sensitive binding sites in cardiac sarcolemma

Dec 15, 1987·Biochemical Pharmacology·J BanningA Abram

Development and characterization of anti-spiroperidol antibodies

Aug 15, 1988·Biochemical Pharmacology·K A Neve, D E Casey

Inhibition of phosphoinositide turnover by selective muscarinic antagonists in the rat striatum. Correlation with receptor occupancy

Jun 15, 1988·Biochemical Pharmacology·F J MonsmaW Hoss

8-Substituted xanthines as antagonists at A1- and A2-adenosine receptors

Oct 1, 1988·Biochemical Pharmacology·K A JacobsonJ W Daly

Lactamimides: a novel chemical class of calcium antagonists with diltiazem-like properties

Aug 1, 1989·Biochemical Pharmacology·M G PalfreymanH I Yamamura

Characteristic beta-adrenergic receptors in a rat ascites hepatoma cell line (AH130)

Oct 15, 1989·Biochemical Pharmacology·K MiyamotoR Koshiura

Iloprost binding and inhibition of aggregation in platelet rich plasma. Differences between normal and type IIa hypercholesterolemic subjects

Jan 1, 1989·Biochemical Pharmacology·D W OlivaE Tremoli

125I-iodopindolol binding to frog esophageal peptic cells. Detection of amine uptake and beta-adrenergic receptors coupled to pepsinogen secretion

May 1, 1989·Biochemical Pharmacology·K E DickinsonB I Hirschowitz

Inhibition of dopamine beta-hydroxylase by captopril

Mar 15, 1989·Biochemical Pharmacology·P PalatiniP Finotti

Pharmacology of binding of 3H-SCH-23390 to D-1 dopaminergic receptor sites in rat striatal tissue

Feb 1, 1989·Biochemical Pharmacology·G FaeddaR J Baldessarini

Nicotine antagonists: phosphoinositide turnover and receptor binding to determine muscarinic properties

Sep 1, 1989·Biochemical Pharmacology·S Benerjee, L G Abood

Characterization of platelet thromboxane A2/prostaglandin H2 receptor by a novel thromboxane receptor antagonist, [3H]S-145

Jun 15, 1989·Biochemical Pharmacology·K HanasakiH Arita

Interaction of fluoxetine with the human placental serotonin transporter

Nov 1, 1990·Biochemical Pharmacology·D R CoolV Ganapathy

Characterization of the beta-adrenergic transduction system in spleen mononuclear leukocyte membranes of young and senescent rats

Jun 15, 1990·Biochemical Pharmacology·P VanscheeuwijckN Fraeyman

Muscarinic receptor antagonist activity of diacylglycerol lipase and kinase inhibitors

Jun 15, 1990·Biochemical Pharmacology·M C SekarL E Hokin

Characterization of cyclic nucleotide phosphodiesterases from cultured bovine aortic endothelial cells

Jan 1, 1990·Biochemical Pharmacology·C Lugnier, V B Schini

Inhibition of muscarinic cholinergic receptors by disulfide reducing agents and arsenicals. Differential effect on locust and rat

Mar 1, 1991·Biochemical Pharmacology·M I FonsecaJ S Aguilar

Muscarinic receptors in diabetic rat prostate

Dec 11, 1991·Biochemical Pharmacology·J LatifpourR M Weiss

The role of enzyme and substrate concentration in the evaluation of serum angiotensin converting enzyme (ACE) inhibition by enalaprilat in vitro

Oct 9, 1991·Biochemical Pharmacology·K Weisser, J Schloos

Interactions of chloroquine with benzodiazepine, gamma-aminobutyric acid and opiate receptors

May 15, 1991·Biochemical Pharmacology·L LiuM Gavish

The relationship between the occupation of the D-1 dopamine receptor by [3H]piflutixol and the activity of dopamine-sensitive adenylate cyclase in rat striatal membranes

Jul 5, 1991·Biochemical Pharmacology·S Fleminger

Delta opioid receptor radioligands

Nov 3, 1992·Biochemical Pharmacology·R J Knapp, H I Yamamura

Characterization of muscarinic cholinergic receptors in intact myocardial cells in vitro

Jun 9, 1992·Biochemical Pharmacology·M Waisberg, A Shainberg

Binding characteristics of the new thromboxane A2/prostaglandin H2 receptor antagonist [3H]BAY U 3405 to washed human platelets and platelet membranes

Aug 4, 1992·Biochemical Pharmacology·J G TheisR Gross

Absence of a direct coupling of a G protein to dihydropyridine binding sites in rat heart

Oct 20, 1992·Biochemical Pharmacology·F HuguetC Dubray

Homoanatoxin: a potent analogue of anatoxin-A

Feb 4, 1992·Biochemical Pharmacology·S WonnacottT Gallagher

Agonist activity of 2- and 5'-substituted adenosine analogs and their N6-cycloalkyl derivatives at A1- and A2-adenosine receptors coupled to adenylate cyclase

Mar 3, 1992·Biochemical Pharmacology·J W Daly, W L Padgett

Pharmacological characterization of a beta 3-receptor agonist (BRL 37,344) and a partial agonist (CGP 12,177A) in neonatal rat liver plasma membranes

Dec 15, 1992·Biochemical Pharmacology·N FraeymanP Vanscheeuwijck

Characterization of solubilized bradykinin B2 receptors from smooth muscle and mucosa of guinea pig ileum

Apr 15, 1992·Biochemical Pharmacology·R W RansomC B Goodman

Partial agonist properties of rauwolscine and yohimbine for the inhibition of adenylyl cyclase by recombinant human 5-HT1A receptors

Jun 9, 1993·Biochemical Pharmacology·J M ArthurJ R Raymond

Binding of [3H]SR 27417, a novel platelet-activating factor (PAF) receptor antagonist, to rabbit and human platelets and polymorphonuclear leukocytes

Jan 7, 1993·Biochemical Pharmacology·J M HerbertJ P Maffrand

Species-dependent differences in the biochemical effects and metabolism of 5-benzylacyclouridine

Jan 7, 1993·Biochemical Pharmacology·S T DavisD P Baccanari

Metabolism and mode of selective inhibition of human immunodeficiency virus replication by 3'-azido-2',3'-dideoxy-5-iodouridine and 3'-azido-2',3'-dideoxy-5-bromouridine

Jan 7, 1993·Biochemical Pharmacology·E M AugustW H Prusoff

Translocation of dopamine and binding of 2 beta-carbomethoxy-3 beta-(4-fluorophenyl) tropane (WIN 35,428) measured under identical conditions in rat striatal synaptosomal preparations. Inhibition by various blockers

Jan 31, 1995·Biochemical Pharmacology·C XuM E Reith

5-Isothiocyanonicotine: a high-affinity irreversible ligand for brain nicotinic receptors

Jun 1, 1994·Biochemical Pharmacology·K D KimL G Abood

Malformin-A1 inhibits the binding of interleukin-1 beta (IL1 beta) and suppresses the expression of tissue factor in human endothelial cells and monocytes

Sep 15, 1994·Biochemical Pharmacology·J M HerbertX Emonds-Alt

Methadone: a potent inhibitor of rat liver aldehyde oxidase

Feb 9, 1994·Biochemical Pharmacology·I G Robertson, R S Gamage

Binding characteristics of the adenosine A2 receptor ligand [3H]CGS 21680 to human platelet membranes

Oct 18, 1994·Biochemical Pharmacology·K VaraniE Ongini

Inhibition of spinal noradrenaline uptake in rats by the centrally acting analgesic tramadol

Jun 15, 1994·Biochemical Pharmacology·W Reimann, H H Hennies

Pharmacological characterization of linear analogues of vasopressin generated by the systematic substitution of positions 1 and 6 by L-amino acids

Apr 29, 1994·Biochemical Pharmacology·J HowlM Wheatley

The intracellular phosphorylation of (-)-2'-deoxy-3'-thiacytidine (3TC) and the incorporation of 3TC 5'-monophosphate into DNA by HIV-1 reverse transcriptase and human DNA polymerase gamma

Sep 28, 1995·Biochemical Pharmacology·N M GrayR C Bethell

Effects of halothane on the nicotinic acetylcholine receptor from Torpedo californica

Apr 18, 1995·Biochemical Pharmacology·L LinH Wang

Effects of propofol and thiopentone on potassium- and carbachol-evoked [3H]noradrenaline release and increased [Ca2+]i from SH-SY5Y human neuroblastoma cells

Jun 28, 1996·Biochemical Pharmacology·D G LambertG Smith

Alpha 1-adrenergic receptors and stimulation of [3H]inositol metabolism in rat brain: regional distribution and parallel inactivation

Aug 19, 1985·Brain Research·R D Johnson, K P Minneman

Binding of [3H]Ro 5-4864 in primary cultures of astrocytes

Aug 19, 1985·Brain Research·A S Bender, L Hertz

Muscarinic cholinergic receptor subtypes in the human brain. II. Quantitative autoradiographic studies

Jan 8, 1986·Brain Research·R CortésJ M Palacios

Measurement and characterization of neuronal cholecystokinin using a novel radioreceptor assay

Nov 29, 1986·Brain Research·I J BeresfordJ Hughes

Changes in cortical beta-adrenergic receptor density and neuronal sensitivity to norepinephrine accompany morphine dependence and withdrawal

Jan 1, 1987·Brain Research·H C Moises, C B Smith

Muscarinic M2 receptor-mediated cyclic AMP reduction in mechanically dissociated rat cortex

Dec 13, 1988·Brain Research·D J Anderson, M McKinney

Correlation of ontogeny with function of [3H]U69593 labelled kappa opioid binding sites in the rat spinal cord

Nov 13, 1989·Brain Research·C A AllertonJ Hughes

Characterization of [125I]HEAT binding to alpha 1-receptors in human brain: assessment in aging and Alzheimer's disease

Nov 6, 1989·Brain Research·R N Kalaria

Electrophysiological responsiveness to isoproterenol in rat hippocampal slices correlates with changes in beta-adrenergic receptor density induced by chronic morphine treatment

Apr 17, 1989·Brain Research·H C Moises, C B Smith

Characterization of zeta (zeta): a new opioid receptor involved in growth

Mar 20, 1989·Brain Research·I S ZagonP J McLaughlin

Evidence for multiple [3H]prazosin binding sites in canine brain membranes

May 1, 1989·Brain Research·E MignotR Ciaranello

Localization and characterization of somatostatin binding sites in the mouse retina

Jan 2, 1989·Brain Research·M KossutL H Pinto

Adrenal steroid type I and type II receptor binding: estimates of in vivo receptor number, occupancy, and activation with varying level of steroid

Apr 23, 1990·Brain Research·R L SpencerB S McEwen

Characterization of oxytocin-binding sites in primary rat brain cell cultures

Jul 30, 1990·Brain Research·D Di Scala-GuenotP Richard

Specific binding of resiniferatoxin, an ultrapotent capsaicin analog, by dorsal root ganglion membranes

Jul 30, 1990·Brain Research·A Szallasi, P M Blumberg

D1 dopamine receptors in neurite regions of embryonic and differentiated retina are highly coupled to adenylate cyclase in the embryonic but not in the mature tissue

Oct 22, 1990·Brain Research·A L Ventura, F G de Mello

The binding of somatostatin to the mouse retina is altered by the pearl mutation

Jul 9, 1990·Brain Research·M KossutL H Pinto

Differential effects of DSP-4 on noradrenaline axons in cerebral cortex and hypothalamus may reflect heterogeneity of noradrenaline uptake sites

Jul 9, 1990·Brain Research·R ZaczekR Grzanna

XAMI and DCDM, agonists at cAMP-associated octopamine receptors in cockroach nerve cord, produce centrally mediated antinociception in mice

Sep 20, 1991·Brain Research·R B RaffaR M Hollingworth

Rods and cones activate different excitatory amino acid receptors on the mudpuppy retinal horizontal cell

Jan 4, 1991·Brain Research·H G Kim, R F Miller

Characterization of muscarinic receptor subtype of rat eccrine sweat gland by autoradiography

May 31, 1991·Brain Research·N E TorresP A Low

Chronic exposure to delta 9-tetrahydrocannabinol fails to irreversibly alter brain cannabinoid receptors

Apr 1, 1991·Brain Research·T M WestlakeW Slikker

Zeta (zeta), a growth-related opioid receptor in developing rat cerebellum: identification and characterization

Jun 14, 1991·Brain Research·I S ZagonP J McLaughlin

Autoradiographic visualization and characteristics of [125I]bradykinin binding sites in guinea pig brain

Apr 10, 1992·Brain Research·P J PriviteraC R Hiley

Galanin receptors from human pituitary tumors assayed with human galanin as ligand

Oct 15, 1993·Brain Research·A L HultingT Bartfai

Long-lasting decrease in dopamine uptake sites following repeated administration of methamphetamine in the rat striatum

Jan 22, 1993·Brain Research·M NakayamaI Yamashita

Subtype-specificity of the presynaptic alpha 2-adrenoceptors modulating hippocampal norepinephrine release in rat

Mar 20, 1995·Brain Research·J P KissE S Vizi

Interactions between laudanosine, GABA, and opioid subtype receptors: implication for laudanosine seizure activity

May 23, 1994·Brain Research·Y KatzM Gavish

Identification of endothelin receptor subtypes in rat retina using subtype-selective ligands

Aug 28, 1995·Brain Research·J A de JuanR Fernandez-Durango

A practical computer-based approach to the analysis of radioligand binding experiments

Aug 1, 1983·Computer Programs in Biomedicine·G A McPherson

Tricyclic antidepressive drugs and dopamine-sensitive adenylate cyclase from rat brain striatum

Feb 1, 1975·European Journal of Pharmacology·M E Karobath

Regional effects of neuroleptics on dopamine metabolism and dopamine-sensitive adenylate cyclase activity

Aug 15, 1977·European Journal of Pharmacology·B ScattonJ Korf

Nomifensine and its derivatives as possible tools for studying amine uptake

Mar 21, 1977·European Journal of Pharmacology·J Tuomisto

Opiate receptor binding affected differentially by opiates and opioid peptides

Apr 1, 1979·European Journal of Pharmacology·S R ChildersS H Synder

Opioid activities of fragments of beta-endorphin and of its leucine65-analogue. Comparison of the binding properties of methionine- and leucine-enkephalin

Sep 1, 1979·European Journal of Pharmacology·A A WaterfieldH W Kosterlitz

High affinity binding of tricyclic antidepressants to histamine H1-receptors: fact and artifact

Oct 3, 1980·European Journal of Pharmacology·J E Taylor, E Richelson

Cardiac muscarinic cholinergic receptor sites: opposing regulation by divalent cations and guanine nucleotides of receptor-agonist interaction

Apr 4, 1980·European Journal of Pharmacology·J W Wei, P V Sulakhe

Displacement of [3H]clonidine binding by clonidine analogues in membranes from rat cerebral cortex

Aug 29, 1980·European Journal of Pharmacology·R J SummersW J Louis

Human platelet 5HT receptors: characterisation and functional association

Dec 5, 1980·European Journal of Pharmacology·J R Peters, D G Grahame-Smith

Alpha 2-adrenoreceptors on human platelets: selective labelling by [3H]clonidine and [3H]yohimbine and competitive inhibition by antidepressant drugs

Sep 24, 1981·European Journal of Pharmacology·J A García-SevillaC B Smnith

125I]BE 2254, a new high affinity radioligand for alpha 1-adrenoceptors

Jul 17, 1981·European Journal of Pharmacology·G Engel, D Hoyer

Atypical characteristics of frog and chick erythrocyte beta-adrenoceptors

Aug 27, 1981·European Journal of Pharmacology·K E Dickinson, S R Nahorski

Muscarinic receptor of rat pancreatic acini: [3H]QNB binding and amylase

Dec 3, 1981·European Journal of Pharmacology·L LaroseG G Poirier

Brain histamine H1- and H2-receptors and histamine-sensitive adenylate cyclase: effects of antipsychotics and antidepressants

Sep 11, 1981·European Journal of Pharmacology·J Coupet, V A Szuchs-Myers

Temperature dependence of [3H]dihydroalprenolol binding in rat myocardium

Jan 22, 1982·European Journal of Pharmacology·R Winek, R Bhalla

High-affinity binding of [3H]doxepin to histamine H1-receptors in rat brain: possible identification of a subclass of histamine H1-receptors

Mar 12, 1982·European Journal of Pharmacology·J E Taylor, E Richelson

Specificity of the beta 2-adrenergic receptor stimulating cyclic AMP accumulation in the intermediate lobe of rat pituitary gland

Jul 16, 1982·European Journal of Pharmacology·H Meunier, F Labrie

Interaction of the putative dopamine autoreceptor agonists 3-PPP and TL-99 with [3H]apomorphine binding sites in rat striatal membranes

Dec 17, 1982·European Journal of Pharmacology·M Williams, J A Totaro

In vitro studies with (imidazolinyl-2)-2-benzodioxane-1-4 ((+/-)-170 150), a new potent alpha 2-adrenoceptor blocking agent

Dec 17, 1982·European Journal of Pharmacology·H DabiréP Meyer

Selective labelling of dopamine (D2) receptors in rat striatum by [3H]domperidone but not by [3H]spiperone

Jul 9, 1982·European Journal of Pharmacology·S Lazareno, S R Nahorski

Characterization of (-)-[3H]dihydroalprenolol binding to intact and broken cell preparations of human peripheral blood lymphocytes

Nov 19, 1982·European Journal of Pharmacology·H MeursP L Bruynzeel

Behavioural and biochemical changes following chronic administration of L-dopa to rats

Apr 23, 1982·European Journal of Pharmacology·C PycockC T O'Shaughnessy

Chronic antidepressant treatment enhances agonist affinity of brain alpha 1-adrenoceptors

Jan 28, 1983·European Journal of Pharmacology·D B MenkesD W Gallager

Identification of [3H]prazosin binding sites in crude membranes and isolated cells of brown adipose tissue as alpha 1-adrenergic receptors

Aug 19, 1983·European Journal of Pharmacology·N MohellB Cannon

Interaction of ergot alkaloids and their combination (co-dergocrine) with alpha-adrenoceptors in the CNS

Sep 30, 1983·European Journal of Pharmacology·R MarksteinW Frick

Quantitative differentiation of alpha- and beta-adrenergic respiratory responses in isolated hamster brown fat cells: evidence for the presence of an alpha 1-adrenergic component

Sep 30, 1983·European Journal of Pharmacology·N MohellB Cannon

The selectivity of some ergot derivatives for alpha 1 and alpha 2-adrenoceptors of rat cerebral cortex

Aug 5, 1983·European Journal of Pharmacology·G A McPherson, P M Beart

Opiate binding sites in bovine retina: evidence for benzomorphan selective binding sites

Jan 21, 1983·European Journal of Pharmacology·H H Osborne, A Herz

Inhibitory effects of pirenzepine on muscarinic stimulation of rat pancreas

Sep 2, 1983·European Journal of Pharmacology·J P DehayeJ Christophe

Antidepressants are weak competitive antagonists of histamine H2 receptors in dissociated brain tissue

Oct 28, 1983·European Journal of Pharmacology·S Kanba, E Richelson

Modulation of rat pancreatic amylase secretion and muscarinic receptor populations by chronic bethanechol treatment

Nov 25, 1983·European Journal of Pharmacology·L LaroseJ Morisset

Muscarinic cholinoceptors in the rabbit's myometrium: a study of the relationship between binding and response

May 18, 1984·European Journal of Pharmacology·D J Crankshaw

Increased alpha 1-adrenergic receptor density in brown adipose tissue of cold-acclimated rats and hamsters

Nov 27, 1984·European Journal of Pharmacology·A RaasmajaJ Nedergaard

3H]p-Aminoclonidine binding to multiple alpha 2-adrenoceptor sites in homogenates of cat frontal cortex and cat spinal cord

Nov 27, 1984·European Journal of Pharmacology·J R Howe, T L Yaksh

The effects of serotonin antagonists in a behavioral despair procedure in mice

Dec 15, 1984·European Journal of Pharmacology·D LuttingerM Perrone

Interactions of vasopressin agonists and antagonists with membrane receptors

Apr 13, 1984·European Journal of Pharmacology·F FahrenholzZ Grzonka

The chemical basis for the blockade of the D-1 dopamine receptor by SCH 23390

Apr 13, 1984·European Journal of Pharmacology·Y ItohJ W Kebabian

Characterization of the leukotriene D4 receptor in guinea-pig lung

Jun 15, 1984·European Journal of Pharmacology·S MongS T Crooke

Dose-dependent effects of prolyl-leucyl-glycinamide on morphine-induced analgesia, tolerance and dependence

Jun 15, 1984·European Journal of Pharmacology·P C Contreras, A E Takemori

Blockade by antidepressants and related compounds of biogenic amine uptake into rat brain synaptosomes: most antidepressants selectively block norepinephrine uptake

Sep 17, 1984·European Journal of Pharmacology·E Richelson, M Pfenning

Lack of correlation between [3H]ouabain binding and Na-K ATPase inhibition in rat aorta

Mar 16, 1984·European Journal of Pharmacology·R C DethR Walsh

Actions of betahistine at histamine receptors in the brain

Apr 23, 1985·European Journal of Pharmacology·J M ArrangJ C Schwartz

Characterization of muscarinic receptors in human submandibular salivary glands

Oct 22, 1985·European Journal of Pharmacology·F MartosF Sanchez de La Cuesta

Alpha 2-adrenoceptor coupling to adenylate cyclase in adrenaline insensitive human platelets

Oct 8, 1985·European Journal of Pharmacology·S S SwartD B Barnett

Activation of alpha 1-adrenoceptors increases [3H]inositol metabolism in rat vas deferens and caudal artery

Oct 8, 1985·European Journal of Pharmacology·A W FoxK P Minneman

Kinetic and pharmacological profiles of the in vitro binding of the potent dopamine agonist [3H]N,N-dipropyl-5,6-dihydroxy-2-aminotetralin to rat striatal membranes

May 28, 1985·European Journal of Pharmacology·T B MulderA S Horn

Estradiol-induced increase of specific [3H]ketanserin binding sites on rat uterine membranes

Feb 5, 1985·European Journal of Pharmacology·S IchidaT Murakami

Stereoselectivity of the histamine H3-presynaptic autoreceptor

Oct 29, 1985·European Journal of Pharmacology·J M ArrangW Schunack

Interaction of amoxapine with muscarinic cholinergic receptors: an in vitro assessment

Jun 7, 1985·European Journal of Pharmacology·J CoupetB Beer

Histamine H1-receptors in the guinea-pig urinary bladder

Aug 7, 1985·European Journal of Pharmacology·M KondoC Tanaka

(+)-[3H]SKF 10,047, (+)-[3H]ethylketocyclazocine, mu, kappa, delta and phencyclidine binding sites in guinea pig brain membranes

Feb 12, 1985·European Journal of Pharmacology·S W Tam

Selective labelling of beta 1-adrenoceptors in rabbit lung membranes by (-)[3H]bisoprolol

Aug 15, 1985·European Journal of Pharmacology·X L WangO E Brodde

Effects of guanine nucleotides and cations on agonist affinity of alpha 1-adrenoceptors in brown adipose tissue

Sep 24, 1985·European Journal of Pharmacology·N Mohell, J Nedergaard

Pharmacological characterization and regional distribution of alpha-noradrenergic binding sites of rat spinal cord

Sep 24, 1985·European Journal of Pharmacology·L T GironS G Crist-Orlando

Autoradiographic localization of benzomorphan binding sites in rat brain

Jul 17, 1985·European Journal of Pharmacology·B J CrainJ O McNamara

Differential effects of adrenergic agonists and phorbol esters on the alpha 1-adrenoceptors of hepatocytes and aorta

Jun 19, 1985·European Journal of Pharmacology·J A García-SáinzB B Hoffman

Characterization of serotonin receptors and lack of effect of antidepressant therapy on monoamine functions in various regions of the rabbit brain

Jul 31, 1986·European Journal of Pharmacology·A SchoupsW De Potter

Possible existence of two mechanisms involved in alpha 1-adrenergic action: effect of Sgd 101/75

Jun 5, 1986·European Journal of Pharmacology·J A García-Sáinz, J L Contreras-Rodríguez

Molecular distinction between calf heart and brain muscarine receptors: different N-ethylmaleimide modulation of agonist binding

Jun 5, 1986·European Journal of Pharmacology·P VanderheydenG Vauquelin

Secoverine is a non-selective muscarinic antagonist on rat heart and brain receptors

Aug 7, 1986·European Journal of Pharmacology·F BrunnerJ Christophe

Differences between central and peripheral rat alpha-adrenoceptors revealed using binuclear ligands

Aug 7, 1986·European Journal of Pharmacology·A AdamsL P Wakelin

Binding and effects of catecholestrogens on adenylate cyclase activity, and adrenoceptors, benzodiazepine and GABA receptors in guinea-pig hypothalamic membranes

Sep 23, 1986·European Journal of Pharmacology·G S EtchegoyenG Pérez-Palacios

Alpha 1- and alpha 2-adrenoceptors in the smooth muscle of male and female rabbit urethra

Feb 11, 1986·European Journal of Pharmacology·F YablonskyJ P Dausse

Stereotyped behavior correlates better than ataxia with phencyclidine-receptor interactions

Feb 11, 1986·European Journal of Pharmacology·P C ContrerasT L O'Donohue

Characterization of alpha 1-adrenoceptors which increase cyclic AMP accumulation in rat cerebral cortex

Oct 7, 1986·European Journal of Pharmacology·R D Johnson, K P Minneman

Enhancement of central and peripheral alpha 1-adrenoceptor sensitivity and reduction of alpha 2-adrenoceptor sensitivity following chronic imipramine treatment in rats

Jan 29, 1986·European Journal of Pharmacology·K W HongW S Lee

Heterogeneity of mammalian alpha 2-adrenoceptors delineated by [3H]yohimbine binding

Jan 29, 1986·European Journal of Pharmacology·K E DickinsonP S Sever

Phosphoinositide hydrolysis mediated by histamine H1-receptors in rat brain cortex

Apr 16, 1986·European Journal of Pharmacology·E ClaroF Picatoste

Alpha-adrenoceptor antagonistic and calcium antagonistic effects of nicergoline in the rat isolated aorta

Apr 16, 1986·European Journal of Pharmacology·C HeitzJ C Stoclet

Dicyclomine, benzhexol and oxybutynine distinguish between subclasses of muscarinic binding sites

Apr 9, 1986·European Journal of Pharmacology·L Nilvebrant, B Sparf

Thermogenic responses to adrenoceptor agonists and brown fat adrenoceptors in overfed rats

Jun 24, 1986·European Journal of Pharmacology·N J RothwellD K Sudera

Phenothiazine drug metabolites: dopamine D2 receptor, alpha 1- and alpha 2-adrenoceptor binding

Jun 24, 1986·European Journal of Pharmacology·P A HalsS G Dahl

Autoradiographic localization and characterization of substance P binding in dog kidney

Oct 27, 1987·European Journal of Pharmacology·J A StephensonE Burcher

Ketanserin blocks alpha 1-adrenoceptors of porcine vascular smooth muscle cells

Jan 13, 1987·European Journal of Pharmacology·J NishimuraM Nakamura

L-652,469--a dual receptor antagonist of platelet activating factor and dihydropyridines from Tussilago farfara L

Sep 11, 1987·European Journal of Pharmacology·S B HwangR J Winquist

Comparison of muscarinic acetylcholine binding in the urinary bladder and submandibular gland of the rabbit

Jun 12, 1987·European Journal of Pharmacology·S Batra

Regulation of high- and low-affinity [3H]imipramine recognition sites in rat brain by chronic treatment with antidepressants

Jun 19, 1987·European Journal of Pharmacology·P D Hrdina

The binding of [3H]leukotriene C4 to guinea-pig lung membranes. The lack of correlation of LTC4 functional activity with binding affinity

Nov 17, 1987·European Journal of Pharmacology·P NormanN J Cuthbert

Pharmacological properties of a proenkephalin A-derived opioid peptide: BAM 18

Jun 26, 1987·European Journal of Pharmacology·D E HurlbutF M Leslie

Identification and characterisation of beta-adrenoceptors in guinea-pig skeletal muscle

Jul 2, 1987·European Journal of Pharmacology·M S Elfellah, J L Reid

Characterization of muscarinic receptors in salivary and lacrimal glands of the rat

Nov 10, 1987·European Journal of Pharmacology·F MartosR Hammer

Muscarinic receptor heterogeneity in guinea pig intestinal smooth muscle: binding studies with AF-DX 116

Sep 23, 1987·European Journal of Pharmacology·E GiraldoR Hammer

Vasopressin receptor mediated contraction and [3H]inositol metabolism in rat tail artery

Mar 3, 1987·European Journal of Pharmacology·A W FoxP W Abel

Functional receptors for fish neuropeptide urotensin II in major rat arteries

Apr 27, 1988·European Journal of Pharmacology·H ItohK Lederis

Selective agents for muscarinic receptors linked to phosphoinositide breakdown

Sep 13, 1988·European Journal of Pharmacology·L Noronha-BlobW J Kinnier

Selectivity of ligand binding to opioid receptors in brain membranes from the rat, monkey and guinea pig

Apr 13, 1988·European Journal of Pharmacology·M J ClarkF Medzihradsky

Muscarinic M1, M2 receptor binding. Relationship with functional efficacy

Oct 26, 1988·European Journal of Pharmacology·S B FreedmanE A Harley

Involvement of the spleen in the endotoxin-induced deterioration of the respiratory airway and lymphocyte beta-adrenergic systems of the guinea pig

Mar 15, 1988·European Journal of Pharmacology·A J Van OosterhoutF P Nijkamp

Characterization of the muscarinic receptor subtypes in the rat urinary bladder

Mar 15, 1988·European Journal of Pharmacology·E MonferiniH Ladinsky

Methoctramine, a polymethylene tetraamine, differentiates three subtypes of muscarinic receptor in direct binding studies

Jan 5, 1988·European Journal of Pharmacology·A Michel, R L Whiting

Regulation of beta-adrenoceptors by catecholamines in the rabbit skeletal muscle

Nov 22, 1988·European Journal of Pharmacology·M S ElfellahJ L Reid

Indolealkylamine analogs share 5-HT2 binding characteristics with phenylalkylamine hallucinogens

Jan 19, 1988·European Journal of Pharmacology·R A LyonR A Glennon

Methoctramine reveals heterogeneity of M2 muscarinic receptors in longitudinal ileal smooth muscle membranes

Jan 19, 1988·European Journal of Pharmacology·A Michel, R L Whiting

Phencyclidine blocks histamine H3-receptors in rat brain

Nov 15, 1988·European Journal of Pharmacology·J M ArrangJ C Schwartz

Adrenoceptor occupancy in isolated human fat cells and its relationship with lipolysis rate

Jan 27, 1988·European Journal of Pharmacology·P ArnerP Engfeldt

Photoaffinity labeling of peripheral-type benzodiazepine receptors in rat kidney mitochondria with [3H]PK 14105

Mar 29, 1988·European Journal of Pharmacology·R SkowrońskiK Beaumont

Antagonism of the responses to isoproterenol in the rat hippocampal slice with subtype-selective antagonists

Aug 9, 1988·European Journal of Pharmacology·J C Fowler, J M O'Donnell

3H]quaternised ICS 205-930 labels 5-HT3 receptor binding sites in rat brain

May 10, 1988·European Journal of Pharmacology·K J WatlingJ Saunders

Characterization of [3H]U46619 binding in pig aorta smooth muscle membranes

Jun 22, 1988·European Journal of Pharmacology·S MiharaT Okabayashi

Further characterization of the myocardial alpha-adrenoceptors mediating positive inotropic effects in the rabbit myocardium

Aug 2, 1988·European Journal of Pharmacology·T HiramotoM Endoh

Characterization of the selectivity, specificity and potency of medetomidine as an alpha 2-adrenoceptor agonist

May 20, 1988·European Journal of Pharmacology·R VirtanenL Nyman

Solubilization and characterization of the kappa-opioid receptor type from guinea-pig cerebellum

May 20, 1988·European Journal of Pharmacology·B FrancésJ C Meunier

Thermodynamic analysis of antagonist and agonist interactions with dopamine receptors

Mar 1, 1988·European Journal of Pharmacology·E P DuarteA P Carvalho

5-HT1B receptors are negatively coupled with adenylate cyclase in rat substantia nigra

Jul 7, 1988·European Journal of Pharmacology·R BouhelalJ Bockaert

5-Methyl-urapidil discriminates between subtypes of the alpha 1-adrenoceptor

Jul 7, 1988·European Journal of Pharmacology·G GrossC Rugevics

Presynaptic and postjunctional muscarinic receptors in dog ileum: binding studies

Nov 28, 1989·European Journal of Pharmacology·P KostkaE E Daniel

Demonstration of alpha 1A- and alpha 1B-adrenoceptor binding sites in human brain tissue

Oct 10, 1989·European Journal of Pharmacology·G GrossH M Mehdorn

The alpha 2-adrenoceptor antagonist SK&F 104078 has high affinity for 5-HT1A and 5-HT2 receptors

Jul 18, 1989·European Journal of Pharmacology·A T KilpatrickM Spedding

Antagonistic actions of S-145 on vascular and platelet thromboxane A2 receptors

Nov 21, 1989·European Journal of Pharmacology·S MiharaM Fujimoto

Receptor binding of fluorinated histidine analogs of thyrotropin-releasing hormone in various regions of the rat brain

May 2, 1989·European Journal of Pharmacology·S VonhofV M Labroo

Alpha 2-adrenoceptor in HT29 human colon adenocarcinoma cell-line: study of [3H](-)-adrenaline binding

Mar 21, 1989·European Journal of Pharmacology·J M SenardH Paris

2-[125I]iodomelatonin labels sites with identical pharmacological characteristics in chicken brain and chicken retina

Mar 21, 1989·European Journal of Pharmacology·M L DubocovichM Mickel

Direct measurement of muscarinic agents in the central nervous system of mice using ex vivo binding

Dec 19, 1989·European Journal of Pharmacology·S B FreedmanS Patel

Thromboxane A2 activates phospholipase C in astrocytoma cells via pertussis toxin-insensitive G-protein

Mar 29, 1989·European Journal of Pharmacology·N NakahataH Nakanishi

Direct labeling of rat M3-muscarinic receptors by [3H]4DAMP

Aug 3, 1989·European Journal of Pharmacology·A MichelR L Whiting

A-69024: a non-benzazepine antagonist with selectivity for the dopamine D-1 receptor

Aug 3, 1989·European Journal of Pharmacology·D J KerkmanJ W Kebabian

Subtypes of nucleoside transport inhibitory sites in heart: a quantitative autoradiographical analysis

Apr 12, 1989·European Journal of Pharmacology·F E Parkinson, A S Clanachan

Muscarinic receptor subtypes in human and guinea pig lung

May 19, 1989·European Journal of Pharmacology·J C Mak, P J Barnes

Intrinsic sympathomimetic activity of beta-adrenoceptor antagonists: down-regulation of cardiac beta 1- and beta 2-adrenoceptors

Nov 7, 1989·European Journal of Pharmacology·C ReithmannK Werdan

Desmethoxyverapamil-sensitive calcium channels in rat portal vein smooth muscle

Aug 22, 1989·European Journal of Pharmacology·G LoirandJ Mironneau

Bretylium tosylate binds preferentially to muscarinic receptors labelled with [3H]oxotremorine M (SH or 'high affinity' receptors) in rat heart and brain cortex

Jan 24, 1989·European Journal of Pharmacology·M GillardJ Christophe

Selective and functional 5-hydroxytryptamine3 receptor antagonism by BRL 43694 (granisetron)

Jan 10, 1989·European Journal of Pharmacology·G J Sanger, D R Nelson

Interaction of DPI 201-106 with cardiac muscarinic receptors

Jan 10, 1989·European Journal of Pharmacology·K GroschnerW R Kukovetz

3H]idazoxan binding at non-alpha 2-adrenoceptors in rabbit adipocyte membranes

Jan 10, 1989·European Journal of Pharmacology·D Langin, M Lafontan

Muscarinic receptor binding characteristics of a human neuroblastoma SK-N-SH and its clones SH-SY5Y and SH-EP1

Jun 8, 1989·European Journal of Pharmacology·D G LambertS R Nahorski

Association of [3H]zacopride with 5-HT3 binding sites

Sep 22, 1989·European Journal of Pharmacology·L M PinkusJ C Gordon

Competitive inhibition of platelet thromboxane A2 receptor binding by picotamide

Oct 4, 1989·European Journal of Pharmacology·P A ModestiG Neri Serneri

UH-AH 37, an ileal-selective muscarinic antagonist that does not discriminate between M2 and M3 binding sites

Feb 28, 1989·European Journal of Pharmacology·H N Doods, N Mayer

Atropine- and scopolamine-resistant subtypes of muscarinic receptors in the rabbit aorta

Dec 12, 1989·European Journal of Pharmacology·S Manjeet, M K Sim

In vivo characterisation of novel efficacious muscarinic receptor agonists

Oct 9, 1990·European Journal of Pharmacology·S B FreedmanS Patel

The anti-aggressive drug eltoprazine preferentially binds to 5-HT1A and 5-HT1B receptor subtypes in rat brain: sensitivity to guanine nucleotides

Oct 9, 1990·European Journal of Pharmacology·H SijbesmaE R De Kloet

Characterization of muscarinic acetylcholine receptors in human labial salivary glands

Feb 13, 1990·European Journal of Pharmacology·L MeiH I Yamamura

High-affinity binding of mequitamium iodide (LG 30435) to muscarinic and histamine H1 receptors

Jul 17, 1990·European Journal of Pharmacology·A R RenzettiM Criscuoli

Pharmacological characterization of melatonin binding sites in Syrian hamster hypothalamus

Jan 3, 1990·European Journal of Pharmacology·D S Pickering, L P Niles

Binding of the cage convulsant, [3H]TBOB, to sites linked to the GABAA receptor complex

Apr 25, 1990·European Journal of Pharmacology·C M Van RijnJ F Rodrigues de Miranda

Metabolites of haloperidol display preferential activity at sigma receptors compared to dopamine D-2 receptors

Feb 27, 1990·European Journal of Pharmacology·W D BowenJ M Walker

The inhibition of [3H]leukotriene D4 binding to guinea-pig lung membranes. The correlation of binding affinity with activity on the guinea-pig ileum

Jul 3, 1990·European Journal of Pharmacology·P NormanP J Gardiner

On the interaction of gallamine with muscarinic receptor subtypes

Jul 3, 1990·European Journal of Pharmacology·A MichelR L Whiting

High-affinity [3H]6-nitroquipazine binding sites in rat brain

May 16, 1990·European Journal of Pharmacology·K Hashimoto, T Goromaru

High-affinity binding of [3H]6-nitroquipazine to 5-hydroxytryptamine transporter in human platelets

Oct 23, 1990·European Journal of Pharmacology·K Hashimoto, T Goromaru

Antagonism of [3H]zacopride binding to 5-HT3 recognition sites by its (R) and (S) enantiomers

Apr 10, 1990·European Journal of Pharmacology·L M PinkusH R Munson

Characterization of kappa-opioid receptors in the guinea-pig ileum

Jun 21, 1990·European Journal of Pharmacology·V U DissanayakeJ Hughes

The binding of [3H]4-diphenylacetoxy-N-methylpiperidine methiodide to longitudinal ileal smooth muscle muscarinic receptors

Feb 6, 1990·European Journal of Pharmacology·A Michel, R L Whiting

Norvaline2-TRH: binding to TRH receptors in rat brain homogenates

May 3, 1990·European Journal of Pharmacology·S VonhofV M Labroo

ONO NT-126 is a potent and selective thromboxane A2 antagonist in human astrocytoma cells

Aug 10, 1990·European Journal of Pharmacology·N NakahataH Nakanishi

Identification of alpha 2-adrenoceptors and non-adrenergic idazoxan binding sites in rabbit colon epithelial cells

Nov 20, 1990·European Journal of Pharmacology·J M SenardH Paris

Carbachol-induced potentiation and inhibition of acid secretion by guinea pig gastric gland

Mar 13, 1990·European Journal of Pharmacology·M KajimuraN Honda

Autoradiographic localization of dopamine receptors in rat cerebral blood vessels

Jan 3, 1991·European Journal of Pharmacology·F AmentaJ A Vega

Cardioselectivity of AQ-RA 741, a novel tricyclic antimuscarinic drug

Jan 3, 1991·European Journal of Pharmacology·H N DoodsN Mayer

3H]ohmefentanyl preferentially binds to mu-opioid receptors but also labels sigma-sites in rat brain sections

Feb 14, 1991·European Journal of Pharmacology·H WangW Rostène

CCK-8-related C-terminal tetrapeptides: affinities for central CCKB and peripheral CCKA receptors

Dec 17, 1991·European Journal of Pharmacology·R HarhammerH Repke

Dopamine D2 receptor binding properties of [3H]U-86170, a dopamine receptor agonist

Sep 17, 1991·European Journal of Pharmacology·R A LahtiR S Hsi

Binding affinity and antimuscarinic activity of sigma and phencyclidine receptor ligands

Mar 19, 1991·European Journal of Pharmacology·H M Vargas, R N Pechnick

The antihypertensive effect of 2-alkynyladenosines and their selective affinity for adenosine A2 receptors

Apr 10, 1991·European Journal of Pharmacology·T AbiruA Matsuda

Dynorphin A-(1-13)-Tyr14-Leu15-Phe16-Asn17-Gly18-Pro19 : a potent and selective kappa opioid peptide

Apr 17, 1991·European Journal of Pharmacology·G P MartinkaS Lemaire

High affinity receptor binding of platelet-activating factor in rat peritoneal polymorphonuclear leukocytes

Apr 17, 1991·European Journal of Pharmacology·S B Hwang

Evaluation of receptor mechanism mediating fentanyl analgesia and toxicity

May 17, 1991·European Journal of Pharmacology·Y Jang, B C Yoburn

Characterization of rat intestinal angiotensin II receptors

Nov 5, 1991·European Journal of Pharmacology·M SchinkeM Entzeroth

Competitive inhibition by NBQX of kainate/AMPA receptor currents and excitatory synaptic potentials: importance of 6-nitro substitution

May 14, 1992·European Journal of Pharmacology·J C RandleJ M Lepagnol

Striatal dopamine D1-like receptors have higher affinity for dopamine in ethanol-treated rats

May 14, 1992·European Journal of Pharmacology·T May

Endocardial localization and characterization of natriuretic peptide binding sites in human fetal and adult heart

Feb 25, 1992·European Journal of Pharmacology·R A RutherfordJ M Polak

Characterization of BIBS 39 and BIBS 222: two new nonpeptide angiotensin II receptor antagonists

Jul 21, 1992·European Journal of Pharmacology·J ZhangJ C Van Meel

Increased density of alpha-adrenoceptors in vas deferens of spontaneously hypertensive rats (SHR), indicated by functional and receptor binding studies

Jul 21, 1992·European Journal of Pharmacology·A Caricati-NetoA Jurkiewicz

Discriminative stimulus properties of the muscarinic receptor agonists Lu 26-046 and O-Me-THPO in rats: evidence for involvement of different muscarinic receptor subtypes

Jul 21, 1992·European Journal of Pharmacology·J ArntH Pedersen

Analgesic potency of TRIMU-5: a mixed mu 2 opioid receptor agonist/mu 1 opioid receptor antagonist

Jun 5, 1992·European Journal of Pharmacology·L A TiveG W Pasternak

A comparison of the selectivities of SCH 23390 with BW737C89 for D1, D2 and 5-HT2 binding sites both in vitro and in vivo

Jan 21, 1992·European Journal of Pharmacology·D R Riddall

Analogues of F8Famide resistant to degradation, with high affinity and in vivo effects

Nov 3, 1992·European Journal of Pharmacology·S GicquelJ M Zajac

Regional distribution and regulation of [125I]calcitonin gene-related peptide binding sites in coronary arteries

Sep 4, 1992·European Journal of Pharmacology·G A KnockJ M Polak

Discovery of a potent atrial natriuretic peptide antagonist for ANPA receptors in the human neuroblastoma NB-OK-1 cell line

Dec 2, 1992·European Journal of Pharmacology·C DelporteJ Christophe

Pulmonary actions of LY255283, a leukotriene B4 receptor antagonist

Nov 23, 1992·European Journal of Pharmacology·S A SilbaughJ H Fleisch

Pancopride, a potent and long-acting 5-HT3 receptor antagonist, is orally effective against anticancer drug-evoked emesis

Nov 10, 1992·European Journal of Pharmacology·A G FernándezD J Roberts

Characterization of BIBN 99: a lipophilic and selective muscarinic M2 receptor antagonist

Sep 21, 1993·European Journal of Pharmacology·H N DoodsW Eberlein

Identification of alpha 1-adrenoceptor subtypes in rat renal proximal tubules

Dec 21, 1993·European Journal of Pharmacology·S M GopalakrishnanM F Lokhandwala

Serotonin-5-O-carboxymethyl-glycyl[125I]tyrosinamide labels the 5-HT1D beta receptor subtype in human cortex

Sep 28, 1993·European Journal of Pharmacology·M S Beer, D N Middlemiss

p-chlorophenylalanine-reversible reduction of sigma binding sites by chronic imipramine treatment in rat brain

Jun 11, 1993·European Journal of Pharmacology·Y ShirayamaK Takahashi

Activity of dihydrothienopyridine S312 enantiomers on L-type Ca2+ channels in isolated rat aorta and cerebral microvessels

Feb 16, 1993·European Journal of Pharmacology·C DessyT Godfraind

CGP 52432: a novel potent and selective GABAB autoreceptor antagonist in rat cerebral cortex

Jun 24, 1993·European Journal of Pharmacology·M LanzaM Raiteri

SR 57227A: a potent and selective agonist at central and peripheral 5-HT3 receptors in vitro and in vivo

Jun 24, 1993·European Journal of Pharmacology·A BachyM Hamon

Characterization of muscarinic receptors in guinea-pig uterus

Dec 7, 1993·European Journal of Pharmacology·H N DoodsM Entzeroth

Comparison of the effects of trimebutine and YM114 (KAE-393), a novel 5-HT3 receptor antagonist, on stress-induced defecation

Dec 7, 1993·European Journal of Pharmacology·K MiyataH Yuki

Topical capsaicin administration protects against trinitrobenzene sulfonic acid-induced colitis in the rat

Nov 9, 1993·European Journal of Pharmacology·C GosoA Szallasi

Selective action of two aporphines at alpha 1-adrenoceptors and potential-operated Ca2+ channels

Feb 9, 1993·European Journal of Pharmacology·M D IvorraM P D'Ocon

Binding of [3H]FH-510 to sigma ligand recognition sites in guinea-pig brain membranes

Jul 6, 1993·European Journal of Pharmacology·M TanakaS Otomo

Characterization of alpha 1-adrenoceptor subtypes in prostate and prostatic urethra of rat, rabbit, dog and man

Nov 16, 1993·European Journal of Pharmacology·R TestaA Leonardi

Pharmacological activity of VUF 9153, an isothiourea histamine H3 receptor antagonist

Nov 30, 1993·European Journal of Pharmacology·J C BarnesC T O'Shaughnessy

A comparison of (-)-deoxybenzomorphans devoid of opiate activity with their dextrorotatory phenolic counterparts suggests role of sigma 2 receptors in motor function

Jan 26, 1993·European Journal of Pharmacology·J M WalkerF I Carroll

Muscarinic M1 receptor agonist actions of muscarinic receptor agonists in rabbit vas deferens

Feb 23, 1993·European Journal of Pharmacology·H E ShannonJ S Ward

3H]p-aminoclonidine and [3H]idazoxan label different populations of imidazoline sites on rat kidney

Feb 23, 1993·European Journal of Pharmacology·A C MacKinnonC M Brown

Age-related changes in Ca2+ channel antagonist receptors in rabbit lower urinary tract

Mar 2, 1993·European Journal of Pharmacology·M YoshidaR M Weiss

Is there a difference in the affinity of histamine H1 receptor antagonists for CNS and peripheral receptors? An in vitro study

Mar 2, 1993·European Journal of Pharmacology·A M Ter LaakH Timmerman

125I]neurokinin A labels pharmacologically distinct populations of NK2 binding sites in hamster and rabbit urinary bladder

Mar 2, 1993·European Journal of Pharmacology·S GuardK J Watling

MPC-1304, another type of dihydropyridine, possessing highly potent vasodilating action

Jul 20, 1993·European Journal of Pharmacology·K MiyoshiM Nagasaka

Defibrotide, a single-stranded polydeoxyribonucleotide acting as an adenosine receptor agonist

Jul 20, 1993·European Journal of Pharmacology·G BianchiG Prino

Autoradiographic localization of [3H]nicardipine binding sites in the human renal artery