Solid-phase parallel synthesis of drug-like artificial 2H-benzopyran libraries.

Molecules : a Journal of Synthetic Chemistry and Natural Product Chemistry
Taeho Lee, Young-Dae Gong

Abstract

This review covers the construction of drug-like 2H-benzopyrans and related libraries using solid-phase parallel synthesis. In this context, the preparation of substituted benzopyrans such as mono-, di- and trisubstituted benzopyran derivatives and additional ring-fused benzopyrans such as benzopyranoisoxazoles, benzopyranopyrazoles, six-membered ring-fused benzopyrans, and polycyclic benzopyrans are highlighted.

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Citations

Jul 31, 2013·ACS Combinatorial Science·Yi-Wen PanWei-Chieh Cheng
Jun 1, 2014·Organic & Biomolecular Chemistry·Nayeon KimYoung-Dae Gong
Apr 23, 2013·Journal of Cancer Research and Clinical Oncology·Seon-Hyeong LeeSoo-Youl Kim
Nov 12, 2015·Molecules : a Journal of Synthetic Chemistry and Natural Product Chemistry·Doohyun LeeTaeho Lee

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