Synthesis of 1-acyl-3-isopropenylbenzimidazolone derivatives and their activity against Botrytis cinerea

Journal of Agricultural and Food Chemistry
Sheng-Kun LiWen-Jun Wu

Abstract

A series of 1-acyl-3-isopropenylbenzimidazolone derivatives were synthesized, and their structures were characterized by (1)H and (13)C NMR and elemental analysis. Their fungicidal activities against Botrytis cinerea were also evaluated by spore germination assay. The acrylic acid, methacrylic acid, 4-chlorophenyl acetic acid, and 2-chlorobenzoic acid derivatives exhibited strong fungicidal activity. This implied that benzimidazolones might be potential fungicide leading compounds.

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Citations

Mar 27, 2012·Journal of Agricultural and Food Chemistry·Jun-Tao FengXing Zhang
Jan 1, 2010·Acta Crystallographica. Section E, Structure Reports Online·Asmaa SaberSeik Weng Ng
Jan 26, 2016·Molecules : a Journal of Synthetic Chemistry and Natural Product Chemistry·Yongling WuXing Zhang
Apr 23, 2016·Molecules : a Journal of Synthetic Chemistry and Natural Product Chemistry·Guang OuyangYuxin He
Nov 1, 2016·Journal of Agricultural and Food Chemistry·Yuhui Bi, Zhiguo Yu
Mar 28, 2013·International Journal of Molecular Sciences·Nan XuZhiqin Ji
May 19, 2012·International Journal of Molecular Sciences·Shaopeng WeiZhiqin Ji

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