Synthesis of functionalized tryptamines by Brønsted acid catalysed cascade reactions

Chemical Communications : Chem Comm
Nicola MelisAngelo Frongia

Abstract

An original synthetic protocol has been developed for the preparation of highly functionalized tryptamines from 2-hydroxycyclobutanone and secondary arylamines via a solvent-free Brønsted acid catalysed two-step reaction sequence.

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Citations

Mar 8, 2016·Organic & Biomolecular Chemistry·Alberto LuridianaFrancesco Secci
Jun 11, 2019·Organic & Biomolecular Chemistry·Lorenza GhisuAngelo Frongia
May 1, 2020·Organic & Biomolecular Chemistry·Francesco SecciPier Carlo Ricci
Nov 18, 2018·Chemical Communications : Chem Comm·Stefania PorcuFrancesco Secci
Nov 14, 2018·Organic Letters·Stefania PorcuFrancesco Secci

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