The direct catalytic enantioselective synthesis of protected aryl beta-hydroxy-alpha-amino acids

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The direct catalytic enantioselective synthesis of protected aryl beta-hydroxy-alpha-amino acids

Abstract

References

Biphenomycins A and B, novel peptide antibiotics. I. Taxonomy, fermentation, isolation and characterization

Iron-binding compounds of Mycobacterium avium, M. intracellulare, M. scrofulaceum, and mycobactin-dependent M. paratuberculosis and M. avium.

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Synthesis of 2-fluoro- and 6-fluoro-(2S,3R)-(3,4-dihydroxyphenyl)serine as potential in vivo precursors of fluorinated norepinephrines

An efficient synthesis of (-)-chloramphenicol via asymmetric catalytic aziridination: a comparison of catalysts prepared from triphenylborate and various linear and vaulted biaryls

Lobocyclamide B from Lyngbya confervoides. Configuration and asymmetric synthesis of beta-hydroxy-alpha-amino acids by (-)-sparteine-mediated aldol addition

Total synthesis of exochelin MN and analogues

Direct asymmetric aldol reactions of glycine schiff base with aldehydes catalyzed by chiral quaternary ammonium salts

Stereoselective synthesis of anti-beta-hydroxy-alpha-amino acids through dynamic kinetic resolution

Catalytic enantio- and diastereoselective aldol reactions of glycine-derived silicon enolate with aldehydes: an efficient approach to the asymmetric synthesis of anti-beta-hydroxy-alpha-amino acid derivatives

Citations

Catalytic enantioselective aldol additions of alpha-isothiocyanato imides to alpha-ketoesters

Toward the development of novel pest management agents based upon insect kinin neuropeptide analogues

Enantioselective magnesium-catalyzed transformations

Catalytic asymmetric 1,2-addition of α-isothiocyanato phosphonates: synthesis of chiral β-hydroxy- or β-amino-substituted α-amino phosphonic acid derivatives

Catalytic Asymmetric Direct Aldol Reaction of α-Alkyl Azlactones and Aliphatic Aldehydes

Organocatalyzed enantioselective Michael addition/cyclization cascade reaction of 3-isothiocyanato oxindoles with arylidene malonates

Catalytic enantioselective aldol reactions

Construction of contiguous tetrasubstituted chiral carbon stereocenters via direct catalytic asymmetric aldol and Mannich-type reactions

Enantioselective Michael/cyclization reaction sequence: scaffold-inspired synthesis of spirooxindoles with multiple stereocenters

Catalytic asymmetric Michael addition/cyclization of isothiocyanato oxindoles: highly efficient and versatile approach for the synthesis of 3,2'-pyrrolidinyl mono- and bi-spirooxindole frameworks

Straightforward access to protected syn alpha-amino-beta-hydroxy acid derivatives

Synthesis of 1,2-amino alcohols by sigmatropic rearrangements of 3-(N-tosylamino)allylic alcohol derivatives

Catalytic asymmetric synthesis of spirooxindoles via addition of isothiocyanato oxindoles to aldehydes under dinuclear nickel Schiff base catalysis

Efficient synthesis of beta-hydroxy-alpha-amino acid derivatives via direct catalytic asymmetric aldol reaction of alpha-isothiocyanato imide with aldehydes

Direct-type aldol reactions of fluorenylidene-protected/activated glycine esters with aldehydes for the synthesis of β-hydroxy-α-amino acid derivatives

Catalytic enantioselective oxidative coupling of saturated ethers with carboxylic acid derivatives

3-isothiocyanato oxindoles serving as powerful and versatile precursors to structurally diverse dispirocyclic thiopyrrolidineoxindoles through a cascade Michael/cyclization process with amino-thiocarbamate catalysts

Catalytic enantioselective ring-opening reaction of meso-aziridines with α-isothiocyanato imides

Base-catalyzed direct aldolization of α-alkyl-α-hydroxy trialkyl phosphonoacetates.

Catalytic Asymmetric Formal [3+2] Cycloaddition of 2-Isocyanatomalonate Esters and Unsaturated Imines: Synthesis of Highly Substituted Chiral γ-Lactams

The magnesium(II)-catalyzed asymmetric ketone-ene reaction under solvent-free conditions: stereocontrolled access to enantioenriched trifluoromethyl-substituted compounds

A highly enantioselective four-component reaction for the efficient construction of chiral β-hydroxy-α-amino acid derivatives

Stereocontrolled synthesis of syn-β-Hydroxy-α-amino acids by direct aldolization of pseudoephenamine glycinamide

Construction of contiguous tetrasubstituted chiral carbon stereocenters via direct catalytic asymmetric aldol reaction of alpha-isothiocyanato esters with ketones

Catalytic asymmetric synthesis of alpha-alkylidene-beta-hydroxy esters via dynamic kinetic asymmetric transformation involving Ba-catalyzed direct aldol reaction

Catalytic asymmetric synthesis of alpha-amino acids

Stereoselective synthesis of highly functionalized structures from lactate-derived halo ketones

An Ireland-Claisen approach to beta-alkoxy alpha-amino acids

Catalytic enantioselective synthesis of alpha,beta-diamino acid derivatives

Direct organocatalytic asymmetric aldol reaction of alpha-isothiocyanato imides to alpha-ketoesters under low ligand loading: a doubly stereocontrolled approach to cyclic thiocarbamates bearing chiral quaternary stereocenters

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Organocatalytic direct asymmetric aldol reactions of 3-isothiocyanato oxindoles to ketones: stereocontrolled synthesis of spirooxindoles bearing highly congested contiguous tetrasubstituted stereocenters

Development of the Ireland-Claisen rearrangement of alkoxy- and aryloxy-substituted allyl glycinates

Enantioselective synthesis of anti-β-hydroxy-α-amido esters via transfer hydrogenation

A unique approach to the concise synthesis of highly optically active spirooxazolines and the discovery of a more potent oxindole-type phytoalexin analogue

Catalytic Enantioselective Ring-Opening and Ring-Closing Reactions of 3-Isothiocyanato Oxindoles and N-(2-Picolinoyl)aziridines

Synthesis of α-amino acids based on chiral tricycloiminolactone derived from natural (+)-camphor

NHC-catalyzed enantioselective [2 + 2] and [2 + 2 + 2] cycloadditions of ketenes with isothiocyanates

Core scaffold-inspired stereoselective synthesis of spiropyrazolones via an organocatalytic Michael/cyclization sequence

Access to Anti or Syn 2-Amino-1,3-diol Scaffolds from a Common Decarboxylative Aldol Adduct

Direct catalytic enantioselective Mannich reactions: synthesis of protected anti-alpha,beta-diamino acids

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